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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T68808 11-Dehydrocorticosterone

11-Dehydrocorticosterone is an endogenous mineralocorticoid. It increases Na+/K+-ATPase mRNA expression in vascular smooth muscle cells and inhibits aldosterone action in B. marinus toad bladder tissue in a concentration-dependent manner. 11-Dehydrocorticosterone decreases the sodium/creatine ratio and increases the potassium/creatine ratio in rat urine in a dose-dependent manner in a model of 11β-hydroxysteroid dehydrogenase inhibition induced by carbenoxolone. Chronic administration 11-dehydro...
T81010 Tetrahydro-11-dehydrocorticosterone

Tetrahydro-11-dehydrocorticosterone 是一种抑制11β-HSD(11β-羟类固醇脱氢酶)的化合物。
T61593 11β-HSD1-IN-6

11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs). These enzymes are responsible for catalyzing the conversion of the active glucocorticoids, corticosterone or cortisol, to their respective inactive forms, 11-dehydrocorticosterone (11-DHC) and cortisone. The compound 11β-HSD1-IN-6 specifically targets and inhibits 11β-HSD-1, effectively modulating the interconversion of these glucocorticoids. [1]

化合物

11-Dehydrocorticosterone
Cat.No: T68808
Synonym:
Target:
Tetrahydro-11-dehydrocorticosterone
Cat.No: T81010
Synonym:
Target:
11β-HSD1-IN-6
Cat.No: T61593
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2884 Cortisone

Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone,可的松

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Cortisone (17-Hydroxy-11-dehydrocorticosterone) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。Cortisone 具有消炎和免疫抑制的作用。Cortisone 在高浓度下对 Glucocorticoid 与Glucocorticoid-receptor 的结合具有部分干预作用。

天然产物

Cortisone
Cat.No: T2884
Synonym: Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone,可的松
Target: Glucocorticoid Receptor, Endogenous Metabolite
TargetMol Loading
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