Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1028 |
Moxonidine
莫索尼定,BDF5895,莫索尼啶 |
Imidazoline Receptor | Neuroscience |
Moxonidine (BDF5895) 是咪唑啉受体亚型 1 的选择性激动剂,用作抗高血压药物。 | |||
T40869 |
Moxonidine hydrochloride
BDF5895hydrochloride,盐酸莫索尼定 |
||
Moxonidine Hydrochloride is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent. Target: I1-R Moxonidine Hydrochloride is a centrally acting antihypertensive agent. Mixed Nischarin (I1 imidazoline receptor) and α2-AR (adrenergic) agonist; displays 40-fold higher affinity for I1 receptors versus α2-adrenoceptors. Moxonidine reduced stimulated NE overflow (log EC50: -6.15 +/- 0.14). AGN192403, a selective ligand at I1-R, had no influence on the dose-response... |