Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0209 |
Ailanthone
臭椿酮,Δ13-Dehydrochaparrinone |
Androgen Receptor | Endocrinology/Hormones |
Ailanthone (Δ13-Dehydrochaparrinone) 是一种有效的雄激素受体 (androgen receptor (AR)) 抑制剂,能够抑制完整雄激素受体(IC50:69 nM)、持续活跃剪切变体(IC50:309 nM)。 |