Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2048L |
α-helical CRF 9-41 acetate
肾上腺皮质素释放因子多肽α-helical CRF 9-41乙酸盐,α-helical CRF 9-41 acetate(90880-23-2 Free base) |
CRFR | GPCR/G Protein |
α-helical CRF 9-41 acetate 是 CRF2 的竞争性拮抗剂 (KB = 100 nM) 和 CRF1 的部分激动剂 (EC50 = 140 nM)。 | |||
TP2048 |
α-Helical CRF(9-41)
α-helical CRF 9-41 |
||
Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively). |