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Cat. No. Product Name Target Signaling Pathways
T80697 β5i-IN-1

Proteasome Proteases/Proteasome; Ubiquitination
β5i-IN-1β5i 选择性抑制剂,具有 8.463 nM 的 IC50 值。该化合物能够诱导 TNF-α 和 IL-6 的释放,同时影响 NF-κB 的转录活性,适用于特发性肺纤维化研究。
T82529 DPLG3

DPLG3是一种免疫蛋白酶体β5i亚基的特异性抑制剂,其对小鼠i-20S的IC50值为9.4 nM,可应用于免疫疾病相关研究领域。
T37420 Ac-ANW-AMC

Ac-ANW-AMC,Ac-Ala-Asn-Trp-AMC

Ac-ANW-AMC is a fluorogenic substrate for the β5i/LMP7 subunit of the 20S immunoproteasome. [1] Upon cleavage, 7-amino-4-methylcoumarin (AMC) is released and its fluorescence can be used to quantify the activity of the β5i/LMP7 subunit of the 20S immunoproteasome. AMC displays excitation/emission maxima of 340-360/440-460 nm, respectively. Reference[1]. Winter, M.B., La Greca, F., Arastu-Kapur, S., et al. Immunoproteasome functions explained by divergence in cleavage specificity and regulation. ...

化合物

β5i-IN-1
Cat.No: T80697
Synonym:
Target: Proteasome
DPLG3
Cat.No: T82529
Synonym:
Target:
Ac-ANW-AMC
Cat.No: T37420
Synonym: Ac-ANW-AMC,Ac-Ala-Asn-Trp-AMC
Target:
TargetMol Loading
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