Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T61519 | α-Glucosidase-IN-18 | ||
α-Glucosidase-IN-18 (7B) is an orally active inhibitor of α-glucosidase, displaying an IC 50 value of 3.96 μM. This compound exhibits antidiabetic properties [1]. | |||
T78740 |
α-Glucosidase-IN-28
|
Glucosidase | Metabolism |
α-Glucosidase-IN-28(Compound 18)是一种有效的α-Glucosidase抑制剂,具有IC50为0.62 μM和Ki为3.93μM。该化合物通过与α-Glucosidase的OBS区域结合以及与周围氨基酸建立多重疏水作用力,展现抑制活性。它主要用于研究糖尿病及其相关疾病。 | |||
T27050 |
CM-10-18
CM-1018 |
||
CM-10-18 is a potent inhibitor of ER α-glucosidase. CM-10-18 demonstrated superior in vitro antiviral activity against representative viruses from four viral families causing hemorrhagic fever. CM-10-18 efficiently protected the lethality of dengue virus |