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Cat. No. | Product Name | Target | Signaling Pathways |
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T72828 |
α-Amylase-IN-2
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α-Glucosidase-IN-3是一种针对α-葡萄糖苷酶(IC50=1.28 µM)和α-淀粉酶(IC50=3.8 µM)的齐墩果酸肟酯衍生物。 | |||
T61706 |
α-Amylase/α-Glucosidase-IN-2
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α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM and 13.09 μM, respectively. This compound shows promise for investigating diabetic complications [1]. | |||
T37835 |
2-Chloro-4-nitrophenyl-α-D-glucopyranoside
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Carbohydrates conjugated with 2-chloro-4-nitrophenyl (CNP) serve as chromogenic substrates in assays for enzymes that release CNP from the conjugated carbohydrate. For example, CNP-β-D-maltoheptaoside and CNP-α-maltotrioside are chromogenic substrates for α-amylase. 2-Chloro-4-nitrophenyl-α-D-glucopyranoside is a conjugate of CNP and α-D-glucose. The related conjugate between CNP and β-D-glucose, 2-chloro-4-nitrophenyl β-D-glucopyranoside, is used as a chromogenic substrate for glycosyltransfera... |
Cat. No. | Product Name | Target | Signaling Pathways |
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T5690 |
7,4'-Di-O-methylapigenin
芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE |
Amylase | Metabolism |
7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) 可能具有抗真菌c.zeyheri 的作用,是一种潜在的抗真菌药物。它还能抑制药物流出泵(IC50 = 51.64μg /毫升)。 | |||
T3S0013 |
Ethyl trans-caffeate
咖啡酸乙酯,Ethyl caffeate,Caffeic Acid Ethyl Ester |
Others | Others |
Ethyl trans-caffeate (Caffeic Acid Ethyl Ester) 具有抗炎作用。 它是一种有前途的天然化合物,未来在慢性肝病中的应用。它是一种有效的化学预防化合物,可防止因太阳紫外线照射引起的皮肤癌变。它是与人胰腺α-淀粉酶复合的代表性抑制剂的高分辨率结构。 它强烈抑制 JB6 Cl41细胞的肿瘤转化,无毒性。 PI3K、ERK1/2 和 p38 激酶活性在体外通过与 HOEC 直接结合而受到抑制。 |