Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1928L1 |
[Orn5]-URP acetate
[Orn5]-URP acetate(782485-03-4 free base) |
GPR | Endocrinology/Hormones; GPCR/G Protein |
[Orn5]-URP acetate 是一种有效的选择性 Urotensin-II receptor (UT) 拮抗剂 (pEC50 = 7.24)。 [Orn5]-URP 没有激动剂活性。 | |||
TP1928 |
[Orn5]-URP
|
||
Urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay. |