Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12660 | (Rac)-BAY1238097 | Epigenetic Reader Domain | Chromatin/Epigenetic |
(Rac)-BAY1238097 is a inhibitor of BET(IC50 of 1.02 μM for BRD4),used in cancer research. | |||
T12660L |
BAY1238097
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
BAY1238097 是一种具有有效性和选择性的溴结构域和末端外基序(BET)抑制剂,具有抗癌活性,在AML (急性髓性白血病) 和MM (多发性骨髓瘤) 模型中表现出较强的抗增殖活性 。BAY1238097 可用于研究晚期难治性恶性肿瘤。 | |||
T13442 | (R)-BAY1238097 | Others | Others |
(R)-BAY1238097 is the R-isomer with lower activity of BAY1238097. BAY1238097 is a selective BET inhibitor. |