Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1960 |
(D)-PPA 1
|
||
PD-1/PD-L1 interaction inhibitor. Binds to PD-L1 (Kd = 0.51 μM). Inhibits interaction at 1 mg/mL in flow cytometry. Inhibits tumor growth and prolongs survival time of mice in vivo. | |||
T78222 |
(D)-PPA 1 TFA
|
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
(D)-PPA 1 TFA为一种抗水解D肽拮抗剂,同时也是有效的PD-1/PD-L1抑制剂。该化合物与PD-1结合亲和力达0.51 μM,且在体内外实验中表现有效。 |