Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22482 |
(±)-Nipecotic acid
|
Others | Others |
(±)-Nipecotic acid is a GABA uptake inhibitor. | |||
T20114 |
Nipecotic acid, S(+)-
(S)-Nipecotic acid,J423.228C,S(+)-nipecotic acid,L-beta-Homoproline |
Others | Others |
Nipecotic acid, S(+)- is an inhibitor of GABA uptake. | |||
T7000 |
Tiagabine hydrochloride
NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Tiagabine hydrochloride (NO050328 hydrochloride) 是具有抗惊厥特性的选择性GABA 再摄取抑制剂,在突触体、神经元和神经胶质中,能够抑制 [3H]GABA 的重摄取,IC50值分别为 67、446 和 182 nM。 |