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PDGFR inhibitor kit

Catalog No. CL0071

PDGFR inhibitor kit 包含血小板衍生生长因子受体 PDGFR 抑制剂,PDGF 受体能够促进细胞的趋化、分裂与增殖、机体生长发育、创伤修复,在调控细胞增殖、分化、生长、发育上扮演相当重要的角色,PDGF 及其受体的高表达促进肿瘤生成,PDGFR 基因突变也可导致肿瘤。PDGFR 抑制剂使肿瘤细胞失去能量来源导致细胞凋亡。TargetMol 为您提供48种精选 PDGFR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
PDGFR inhibitor kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T0093LSorafenib284461-73-0464.8310mMApoptosis; Autophagy; c-Kit; Ferroptosis; FLT; PDGFR; Raf; VEGFR
T0097LPazopanib444731-52-6437.5210mMAutophagy; c-Kit; FGFR; PDGFR; VEGFR
T0374LSunitinib557795-19-4398.4710mMApoptosis; Autophagy; c-Kit; FLT; IRE1; Mitophagy; PDGFR; VEGFR
T1452Axitinib319460-85-0386.4710mMc-Kit; PDGFR; VEGFR
T1667Tandutinib387867-13-2562.710mMApoptosis; c-Kit; CSF-1R; FLT; PDGFR; Src
T1777Nintedanib656247-17-5539.6210mMFGFR; FLT; PDGFR; Src; VEGFR
T1792Regorafenib755037-03-7482.8210mMAutophagy; c-Kit; c-RET; PDGFR; Raf; VEGFR
T1836AZD2932883986-34-3447.4910mMc-Kit; FLT; PDGFR; VEGFR
T2070Agerafenib1188910-76-0517.4610mMBcr-Abl; c-Kit; c-RET; PDGFR; Raf; Src
T2358ENMD-2076934353-76-1375.4710mMApoptosis; Aurora Kinase; c-RET; FGFR; FLT; PDGFR; Src; VEGFR
T2372Ponatinib943319-70-8532.5610mMAutophagy; Bcr-Abl; c-Kit; FGFR; PDGFR; Src; VEGFR
T2415PP1211092788-83-4319.3610mMApoptosis; Bcr-Abl; Hck; mTOR; PDGFR; Src; VEGFR
T2456Tivozanib475108-18-0454.8610mMEphrin Receptor; PDGFR; VEGFR
T2479Tyrphostin A910537-47-0282.3810mMEGFR; Influenza Virus; PDGFR; VEGFR
T2500Cediranib288383-20-0450.5110mMAutophagy; c-Kit; FLT; PDGFR; VEGFR
T2514Linifanib796967-16-3375.410mMApoptosis; Autophagy; c-Fms; c-Kit; CSF-1R; FLT; PDGFR; VEGFR
T2516Amuvatinib850879-09-3447.5110mMApoptosis; c-Kit; c-Met/HGFR; c-RET; DNA/RNA Synthesis; FLT; PDGFR
T2609Masitinib790299-79-5498.6410mMApoptosis; Bcr-Abl; c-Fms; c-Kit; FAK; FGFR; Hck; PDGFR; Src
T2677Crenolanib670220-88-9443.5410mMAutophagy; FLT; PDGFR
T3463NVP-ACC789300842-64-2405.310mMPDGFR; VEGFR
T3476JI-101900573-88-8466.3410mMEphrin Receptor; PDGFR; VEGFR
T6091CP-673451343787-29-1417.510mMc-Kit; PDGFR; VEGFR
T6166Telatinib332012-40-5409.8310mMc-Kit; PDGFR; VEGFR
T6184Orantinib252916-29-3310.3510mMApoptosis; FGFR; PDGFR; VEGFR
T6230Imatinib152459-95-5493.610mMAutophagy; Bcr-Abl; c-Kit; PDGFR; SARS-CoV
T6479Dovitinib lactate hydrate915769-50-5482.5110mMc-Kit; FGFR; FLT; PDGFR; VEGFR
T6711Tyrphostin AG1296146535-11-7266.2910mMApoptosis; c-Kit; FGFR; FLT; PDGFR
T6920ON1233001357470-29-1429.5210mMAMPK; c-RET; CDK; FGFR; JAK; PDGFR; Src
T5001Nintedanib esylate656247-18-6649.7610mMFGFR; PDGFR; VEGFR
T5109Avapritinib1703793-34-3498.5610mMc-Kit; PDGFR; PDGFR
T5466Tyrosine kinase-IN-1705946-27-6445.5410mMFGFR; FLT; PDGFR; VEGFR
T7394Toceranib Phosphate874819-74-6494.4510mMc-Kit; PDGFR; Tyrosinase; VEGFR
T7945SU14813627908-92-3442.4810mMc-Kit; PDGFR; VEGFR
T8491Vorolanib1013920-15-4439.4810mMPDGFR; VEGFR
T8482Ripretinib1442472-39-0510.3610mMApoptosis; c-Kit; FLT; PDGFR; VEGFR
T8541Lenvatinib mesylate857890-39-2522.9610mMc-Kit; c-RET; FGFR; PDGFR; VEGFR
T10157Regorafénib N-oxyde (M2)835621-11-9498.8110mMc-Kit; c-RET; Drug Metabolite; PDGFR; Raf; VEGFR
T15616JNJ-10198409627518-40-5325.3410mMPDGFR
T16750Rigosertib592542-59-1451.4910mMApoptosis; Bcr-Abl; CDK; FLT; PDGFR; PI3K; PLK; Src
T12145LN-Desethylsunitinib hydrochloride1261432-05-6406.8810mMc-Kit; PDGFR; VEGFR
T8900Seralutinib1619931-27-9469.5510mMPDGFR
TQ0235AC7101351522-04-7562.710mMc-Kit; FLT; PDGFR
T16975TAK-5931005780-62-0445.4710mMPDGFR; VEGFR
T13238Tyrphostin AG1433168835-90-3266.2910mMPDGFR; VEGFR
T35570Chiauranib1256349-48-0435.4710mMVEGFR;PDGFR;c-Kit;Aurora Kinase;c-Fms;FLT
T41003KG5877874-85-6459.4510mMRaf;PDGFR;FLT;c-Kit
T16947SU16f251356-45-3386.4410mMPDGFR
T13824PP58212391-58-7456.3310mMPDGFR;FGFR;Src;p38 MAPK;TNF

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产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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