mTOR inhibitor kit 包含哺乳动物雷帕霉素靶蛋白 mTOR 抑制剂,mTOR 是一种高度保守的Ser/Thr 蛋白激酶,许多疾病的发生发展都与mTOR 信号异常有关,持续过度激活的 mTOR 信号会提高细胞代谢水平的、延长细胞寿命甚至使细胞永生化,这将直接或间接诱发癌症、代谢和衰老有关的疾病,mTOR 抑制剂可以有效延缓或治疗mTOR 过度激活引起的癌症、心血管损伤等疾病。TargetMol 为您提供49种精选mTOR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1537 | Rapamycin | 53123-88-9 | 914.18 | 10mM | Antibiotic; Antifungal; Autophagy; Endogenous Metabolite; mTOR |
T1784 | Everolimus | 159351-69-6 | 958.22 | 10mM | Apoptosis; Autophagy; mTOR |
T1838 | Sapanisertib | 1224844-38-5 | 309.33 | 10mM | Autophagy; mTOR; PI3K |
T1859 | AZD-8055 | 1009298-09-2 | 465.54 | 10mM | Apoptosis; Autophagy; mTOR |
T1861 | Omipalisib | 1086062-66-9 | 505.5 | 10mM | Autophagy; mTOR; PI3K |
T1916 | Apitolisib | 1032754-93-0 | 498.6 | 10mM | Apoptosis; mTOR; PI3K |
T1958 | AZ20 | 1233339-22-4 | 412.51 | 10mM | ATM/ATR; mTOR |
T1961 | Vistusertib | 1009298-59-2 | 462.54 | 10mM | Akt; Apoptosis; Autophagy; mTOR; PI3K; S6 Kinase |
T1970 | Gedatolisib | 1197160-78-3 | 615.73 | 10mM | mTOR; PI3K |
T2145 | Temsirolimus | 162635-04-3 | 1030.29 | 10mM | Apoptosis; Autophagy; mTOR |
T2235 | Dactolisib | 915019-65-7 | 469.54 | 10mM | ATM/ATR; Autophagy; mTOR; PI3K |
T2265 | Bimiralisib | 1225037-39-7 | 411.38 | 10mM | mTOR; PI3K; S6 Kinase |
T2357 | GSK1059615 | 958852-01-2 | 333.36 | 10mM | Apoptosis; mTOR; PI3K |
T2414 | Torkinib | 1092351-67-1 | 308.34 | 10mM | Apoptosis; Autophagy; Mitophagy; mTOR; PI3K |
T2415 | PP121 | 1092788-83-4 | 319.36 | 10mM | Apoptosis; Bcr-Abl; Hck; mTOR; PDGFR; Src; VEGFR |
T2475 | KU-0063794 | 938440-64-3 | 465.54 | 10mM | mTOR |
T2706 | Palomid 529 | 914913-88-5 | 406.43 | 10mM | Apoptosis; mTOR |
T3351 | Onatasertib | 1228013-30-6 | 397.47 | 10mM | Apoptosis; c-Fms; DNA-PK; FLT; mTOR; PI3K |
T3395 | Timosaponin AIII | 41059-79-4 | 740.92 | 10mM | AChE; mTOR |
T3514 | CZ415 | 1429639-50-8 | 459.56 | 10mM | mTOR |
T3541 | CC-115 | 1228013-15-7 | 336.35 | 10mM | DNA-PK; mTOR; PI3K |
T3692 | GNE-477 | 1032754-81-6 | 504.63 | 10mM | mTOR; PI3K |
T3986 | SF2523 | 1174428-47-7 | 371.41 | 10mM | DNA-PK; Epigenetic Reader Domain; mTOR; PI3K |
T6045 | Torin 1 | 1222998-36-8 | 607.62 | 10mM | Autophagy; DNA-PK; mTOR; PI3K |
T6100 | Torin 2 | 1223001-51-1 | 432.4 | 10mM | Apoptosis; ATM/ATR; Autophagy; DNA-PK; mTOR |
T6103 | VS-5584 | 1246560-33-7 | 354.41 | 10mM | mTOR; PI3K |
T6143 | PI-103 | 371935-74-9 | 348.36 | 10mM | Apoptosis; Autophagy; DNA-PK; mTOR; PI3K |
T6251 | PF-04691502 | 1013101-36-4 | 425.48 | 10mM | Akt; Autophagy; mTOR; PI3K |
T6319 | OSI-027 | 936890-98-1 | 406.44 | 10mM | Autophagy; DNA-PK; mTOR; PI3K |
T6334 | Ridaforolimus | 572924-54-0 | 990.21 | 10mM | Autophagy; mTOR |
T6731 | WYE-354 | 1062169-56-5 | 495.53 | 10mM | Apoptosis; Autophagy; mTOR; PI3K |
T6845 | GNE-317 | 1394076-92-6 | 414.48 | 10mM | mTOR; PI3K |
T6883 | Samotolisib | 1386874-06-1 | 406.48 | 10mM | Autophagy; DNA-PK; mTOR; PI3K |
T7014 | Voxtalisib | 934493-76-2 | 270.29 | 10mM | DNA-PK; mTOR; PI3K |
T5338 | mTOR inhibitor-1 | 468747-17-3 | 363.21 | 10mM | Autophagy; mTOR |
T5472 | PQR620 | 1927857-56-4 | 445.48 | 10mM | mTOR |
T7166 | GNE-493 | 1033735-94-2 | 372.44 | 10mM | mTOR; PI3K |
T7343 | PF-04979064 | 1220699-06-8 | 446.5 | 10mM | mTOR; PI3K |
T8569 | DMH-25 | 1685280-21-0 | 489.94 | 10mM | mTOR |
T16567 | PQR530 | 1927857-61-1 | 407.42 | 10mM | mTOR; PI3K |
T11728 | JR-AB2-011 | 329182-61-8 | 398.28 | 10mM | mTOR |
T16355 | NSC781406 | 1676893-24-5 | 627.68 | 10mM | mTOR; PI3K |
T6072L | BGT226 | 915020-55-2 | 534.53 | 10mM | Autophagy; mTOR; PI3K |
T40351 | MHY-1685 | 27406-31-1 | 232.19 | 10mM | mTOR |
T36083 | DS-7423 | 1222104-37-1 | 520.51 | 10mM | mTOR; PI3K |
T10413 | Autogramin-1 | 2375541-73-2 | 485.56 | 10mM | Autophagy; mTOR |
T35343 | MTI-31 | 1567915-38-1 | 474.55 | 10mM | mTOR |
T12459 | PI3K/mTOR Inhibitor-2 | 1848242-58-9 | 478.86 | 10mM | PI3K;mTOR |
T60055 | Chromeceptin | 331859-86-0 | 359.35 | 10mM | IGF-1R;Akt;mTOR |