BET inhibitor kit 包含 BET 抑制剂,BET 抑制剂通过模拟乙酰化的 Lys 结构与 KAc 口袋结合,阻断 BD1或 BD2与 KAc 结合,从而在表观遗传学水平上对基因表达进行调控,可用于白血病、淋巴瘤、乳腺癌、脑瘤和骨髓瘤等的治疗研究。TargetMol 为您提供47种精选BET 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1854 | MS436 | 1395084-25-9 | 383.42 | 10mM | Epigenetic Reader Domain |
T1906 | Molibresib | 1260907-17-2 | 423.9 | 10mM | Epigenetic Reader Domain |
T2072 | BET bromodomain inhibitor | 1505453-59-7 | 445.91 | 10mM | Epigenetic Reader Domain |
T2091 | CPI0610 | 1380087-89-7 | 365.81 | 10mM | c-Myc; Epigenetic Reader Domain |
T2110 | (+)-JQ-1 | 1268524-70-4 | 456.99 | 10mM | Autophagy; Epigenetic Reader Domain; Ligands for Target Protein for PROTAC |
T2120 | I-BET151 | 1300031-49-5 | 415.44 | 10mM | Epigenetic Reader Domain |
T2480 | Apabetalone | 1044870-39-4 | 370.4 | 10mM | Epigenetic Reader Domain; HIV Protease |
T3504 | AZD5153 6-Hydroxy-2-naphthoic acid | 1869912-40-2 | 667.75 | 10mM | Epigenetic Reader Domain |
T3712 | Mivebresib | 1445993-26-9 | 459.47 | 10mM | Apoptosis; Epigenetic Reader Domain |
T4247 | I-CBP112 hydrochloride | 2147701-33-3 | 505 | 10mM | Epigenetic Reader Domain |
T4345 | CeMMEC1 | 440662-09-9 | 336.35 | 10mM | Carboxypeptidase; DNA/RNA Synthesis; Epigenetic Reader Domain |
T4365 | FL-411 | 2118944-88-8 | 341.43 | 10mM | Epigenetic Reader Domain |
T6021 | GSK1324726A | 1300031-52-0 | 434.91 | 10mM | Apoptosis; Epigenetic Reader Domain |
T6032 | Birabresib | 202590-98-5 | 491.99 | 10mM | Epigenetic Reader Domain |
T6173 | BI 2536 | 755038-02-9 | 521.66 | 10mM | Apoptosis; Epigenetic Reader Domain; PLK |
T6222 | PFI-1 | 1403764-72-6 | 347.39 | 10mM | Apoptosis; Autophagy; Epigenetic Reader Domain |
T5362 | Y06036 | 1832671-96-1 | 427.27 | 10mM | Epigenetic Reader Domain |
T5417 | INCB-057643 | 1820889-23-3 | 415.46 | 10mM | Apoptosis; Epigenetic Reader Domain |
T6828 | ZL0420 | 2229039-45-4 | 296.32 | 10mM | Epigenetic Reader Domain |
T7863 | Hexamethylene bisacetamide | 3073-59-4 | 200.28 | 10mM | Epigenetic Reader Domain |
T8495 | Alobresib | 1637771-14-2 | 437.5 | 10mM | Epigenetic Reader Domain |
T19618 | (R)-(-)-JQ1 Enantiomer | 1268524-71-5 | 456.99 | 10mM | Epigenetic Reader Domain |
T17311 | (+)-JQ1 PA | 2115701-93-2 | 437.95 | 10mM | Epigenetic Reader Domain |
TQ0253 | PLX51107 | 1627929-55-8 | 438.48 | 10mM | Epigenetic Reader Domain |
T16154 | MS417 | 916489-36-6 | 414.91 | 10mM | Epigenetic Reader Domain; HIV Protease |
T8601 | 1-benzyl-2-ethyl-4,5,6,7-tetrahydro-1H-indol-4-one | 218934-50-0 | 253.35 | 10mM | Epigenetic Reader Domain |
T8609 | CHEMBRDG-BB 7118966 | 328956-24-7 | 241.09 | 10mM | Epigenetic Reader Domain |
T8658 | NEO2734 | 2081072-29-7 | 435.44 | 10mM | Epigenetic Reader Domain; Histone Acetyltransferase |
T19935 | XD14 | 1370888-71-3 | 421.51 | 10mM | Epigenetic Reader Domain |
T12112 | MS402 | 1672684-68-2 | 370.83 | 10mM | Epigenetic Reader Domain |
T8932 | GSK046 | 2474876-09-8 | 414.48 | 10mM | Epigenetic Reader Domain |
T9020 | GSK620 | 2088410-46-0 | 325.4 | 10mM | Epigenetic Reader Domain |
T9194 | UMB298 | 2266569-73-5 | 479.01 | 10mM | Epigenetic Reader Domain |
T50006 | 3-methyl-1,2,3,4-tetrahydroquinazolin-2-one | 24365-65-9 | 162.19 | 10mM | Epigenetic Reader Domain |
T14776 | BRD4 Inhibitor-10 | 1660117-38-3 | 429.51 | 10mM | Epigenetic Reader Domain |
T15405 | GNE-781 | 1936422-33-1 | 525.59 | 10mM | Epigenetic Reader Domain |
T10521 | ODM-207 | 1801503-93-4 | 375.42 | 10mM | Epigenetic Reader Domain |
T28628 | RVX-297 | 1044871-04-6 | 423.5 | 10mM | Epigenetic Reader Domain |
T9629 | WAY-309060 | 309951-18-6 | 262.26 | 10mM | Epigenetic Reader Domain |
T9703L | GSK778 hydrochloride | T9703L | 548.08 | 10mM | Epigenetic Reader Domain |
T13363 | Y06137 | 2226534-49-0 | 444.57 | 10mM | Epigenetic Reader Domain |
T60072 | ZL0590 | 2230496-99-6 | 512.55 | 10mM | Epigenetic Reader Domain |
T22345 | INCB054329 | 1628607-64-6 | 348.36 | 10mM | Epigenetic Reader Domain; Others |
T13394 | ZEN-3862 | 1952264-33-3 | 340.35 | 10mM | Epigenetic Reader Domain |
T27392 | FT001 | 1778655-51-8 | 467.58 | 10mM | Epigenetic Reader Domain |
T12338 | OXFBD04 | 2231747-03-6 | 296.32 | 10mM | Epigenetic Reader Domain |
T12513 | PNZ5 | 1629277-36-6 | 318.37 | 10mM | Epigenetic Reader Domain |