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BET inhibitor kit

Catalog No. CL0072

BET inhibitor kit 包含 BET 抑制剂,BET 抑制剂通过模拟乙酰化的 Lys 结构与 KAc 口袋结合,阻断 BD1或 BD2与 KAc 结合,从而在表观遗传学水平上对基因表达进行调控,可用于白血病、淋巴瘤、乳腺癌、脑瘤和骨髓瘤等的治疗研究。TargetMol 为您提供47种精选BET 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
BET inhibitor kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T1854MS4361395084-25-9383.4210mMEpigenetic Reader Domain
T1906Molibresib1260907-17-2423.910mMEpigenetic Reader Domain
T2072BET bromodomain inhibitor1505453-59-7445.9110mMEpigenetic Reader Domain
T2091CPI06101380087-89-7365.8110mMc-Myc; Epigenetic Reader Domain
T2110(+)-JQ-11268524-70-4456.9910mMAutophagy; Epigenetic Reader Domain; Ligands for Target Protein for PROTAC
T2120I-BET1511300031-49-5415.4410mMEpigenetic Reader Domain
T2480Apabetalone1044870-39-4370.410mMEpigenetic Reader Domain; HIV Protease
T3504AZD5153 6-Hydroxy-2-naphthoic acid1869912-40-2667.7510mMEpigenetic Reader Domain
T3712Mivebresib1445993-26-9459.4710mMApoptosis; Epigenetic Reader Domain
T4247I-CBP112 hydrochloride2147701-33-350510mMEpigenetic Reader Domain
T4345CeMMEC1440662-09-9336.3510mMCarboxypeptidase; DNA/RNA Synthesis; Epigenetic Reader Domain
T4365FL-4112118944-88-8341.4310mMEpigenetic Reader Domain
T6021GSK1324726A1300031-52-0434.9110mMApoptosis; Epigenetic Reader Domain
T6032Birabresib202590-98-5491.9910mMEpigenetic Reader Domain
T6173BI 2536755038-02-9521.6610mMApoptosis; Epigenetic Reader Domain; PLK
T6222PFI-11403764-72-6347.3910mMApoptosis; Autophagy; Epigenetic Reader Domain
T5362Y060361832671-96-1427.2710mMEpigenetic Reader Domain
T5417INCB-0576431820889-23-3415.4610mMApoptosis; Epigenetic Reader Domain
T6828ZL04202229039-45-4296.3210mMEpigenetic Reader Domain
T7863Hexamethylene bisacetamide3073-59-4200.2810mMEpigenetic Reader Domain
T8495Alobresib1637771-14-2437.510mMEpigenetic Reader Domain
T19618(R)-(-)-JQ1 Enantiomer1268524-71-5456.9910mMEpigenetic Reader Domain
T17311(+)-JQ1 PA2115701-93-2437.9510mMEpigenetic Reader Domain
TQ0253PLX511071627929-55-8438.4810mMEpigenetic Reader Domain
T16154MS417916489-36-6414.9110mMEpigenetic Reader Domain; HIV Protease
T86011-benzyl-2-ethyl-4,5,6,7-tetrahydro-1H-indol-4-one218934-50-0253.3510mMEpigenetic Reader Domain
T8609CHEMBRDG-BB 7118966328956-24-7241.0910mMEpigenetic Reader Domain
T8658NEO27342081072-29-7435.4410mMEpigenetic Reader Domain; Histone Acetyltransferase
T19935XD141370888-71-3421.5110mMEpigenetic Reader Domain
T12112MS4021672684-68-2370.8310mMEpigenetic Reader Domain
T8932GSK0462474876-09-8414.4810mMEpigenetic Reader Domain
T9020GSK6202088410-46-0325.410mMEpigenetic Reader Domain
T9194UMB2982266569-73-5479.0110mMEpigenetic Reader Domain
T500063-methyl-1,2,3,4-tetrahydroquinazolin-2-one24365-65-9162.1910mMEpigenetic Reader Domain
T14776BRD4 Inhibitor-101660117-38-3429.5110mMEpigenetic Reader Domain
T15405GNE-7811936422-33-1525.5910mMEpigenetic Reader Domain
T10521ODM-2071801503-93-4375.4210mMEpigenetic Reader Domain
T28628RVX-2971044871-04-6423.510mMEpigenetic Reader Domain
T9629WAY-309060309951-18-6262.2610mMEpigenetic Reader Domain
T9703LGSK778 hydrochlorideT9703L548.0810mMEpigenetic Reader Domain
T13363Y061372226534-49-0444.5710mMEpigenetic Reader Domain
T60072ZL05902230496-99-6512.5510mMEpigenetic Reader Domain
T22345INCB0543291628607-64-6348.3610mMEpigenetic Reader Domain; Others
T13394ZEN-38621952264-33-3340.3510mMEpigenetic Reader Domain
T27392FT0011778655-51-8467.5810mMEpigenetic Reader Domain
T12338OXFBD042231747-03-6296.3210mMEpigenetic Reader Domain
T12513PNZ51629277-36-6318.3710mMEpigenetic Reader Domain

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产品应用

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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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