p53 inhibitor/reactivator kit 包含p53抑制剂/复活剂,p53是一种肿瘤抑制基因,能与DNA 特异结合,控制着细胞周期的启动。但如果p53基因发生了突变,则对细胞的增殖失去控制,导致细胞癌变,在所有恶性肿瘤中,50%以上会出现p53的突变。TargetMol 为您提供27种精选p53抑制剂/复活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1493 | BH3I-1 | 300817-68-9 | 400.31 | 10mM | Bcl; E1/E2/E3 Enzyme; MDM-2/p53 |
T1798 | RITA | 213261-59-7 | 292.37 | 10mM | Autophagy; DNA Alkylator/Crosslinker; MDM-2/p53; Mdm2; p53 |
T1887 | Inauhzin | 309271-94-1 | 469.58 | 10mM | MDM-2/p53; Sirtuin |
T1919 | Tenovin-1 | 380315-80-0 | 369.48 | 10mM | Autophagy; Dehydrogenase; MDM-2/p53; Mdm2; p53; Sirtuin |
T2158 | Nutlin-3 | 548472-68-0 | 581.49 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53 |
T2243 | Serdemetan | 881202-45-5 | 328.42 | 10mM | Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53; Mdm2; p53 |
T2464 | NSC319726 | 71555-25-4 | 234.32 | 10mM | MDM-2/p53; p53 |
T2707 | Pifithrin-α hydrobromide | 63208-82-2 | 367.3 | 10mM | Aryl Hydrocarbon Receptor; Ferroptosis; MDM-2/p53; p53 |
T3637 | Pifithrin-β hydrobromide | 511296-88-1 | 349.29 | 10mM | Ferroptosis; MDM-2/p53; p53 |
T3798 | Ziyuglycoside I | 35286-58-9 | 766.97 | 10mM | Apoptosis; MDM-2/p53 |
T6023 | Nutlin-3a | 675576-98-4 | 581.49 | 10mM | Apoptosis; Autophagy; E1/E2/E3 Enzyme; MDM-2/p53 |
T6149 | YH239-EE | 1364488-67-4 | 504.41 | 10mM | Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53 |
T6210 | Pifithrin-μ | 64984-31-2 | 181.21 | 10mM | Autophagy; HSP; MDM-2/p53; p53 |
T6254 | Idasanutlin | 1229705-06-9 | 616.48 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T6614 | Nutlin-3b | 675576-97-3 | 581.49 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T6909 | NSC348884 | 81624-55-7 | 636.81 | 10mM | Apoptosis; p53 |
T6954 | PRIMA-1 | 5608-24-2 | 185.22 | 10mM | Apoptosis; Autophagy; Ferroptosis; MDM-2/p53 |
T6965 | RG7112 | 939981-39-2 | 727.78 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T5S0331 | Isoliquiritin | 5041-81-6 | 418.39 | 10mM | Antifungal; p53 |
T8774 | MS7972 | 352553-42-5 | 227.26 | 10mM | Epigenetic Reader Domain; MDM-2/p53 |
T12472 | Pifithrin-α, p-Nitro, Cyclic | 60477-38-5 | 299.35 | 10mM | MDM-2/p53; p53 |
T9129 | Benzonitrile, 3,3'-[(2-oxo-1,3-cyclohexanediylidene)dimethylidyne]bis- (9CI) | 63476-70-0 | 324.38 | 10mM | p53 |
T5555 | Siremadlin | 1448867-41-1 | 555.41 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53 |
TQ0127 | Navtemadlin | 1352066-68-2 | 568.55 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T21578 | NSC 66811 | 6964-62-1 | 340.42 | 10mM | MDM-2/p53 |
T24730 | Roslin 2 bromide | 29574-21-8 | 311.22 | 10mM | p53;FAK |
T27093 | CT-1 | 1983924-33-9 | 500.51 | 10mM | p53 |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |