Histone Demethylase inhibitor kit 包含组蛋白去甲基化酶抑制剂,组蛋白修饰是表观遗传中重要的调控机制之一,组蛋白去甲基化酶在肿瘤的发生发展、个体发育、代谢性疾病如糖尿病等过程中发挥重要作用。TargetMol 为您提供30种精选组蛋白去甲基化酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1025 | Tranylcypromine (2-PCPA) hydrochloride | 1986-47-6 | 169.66 | 10mM | Histone Demethylase; MAO |
T1868 | JIB-04 | 199596-05-9 | 308.76 | 10mM | Apoptosis; Histone Demethylase; Histone Methyltransferase |
T2304 | SP2509 | 1423715-09-6 | 437.9 | 10mM | Apoptosis; Histone Demethylase |
T2315 | GSK-LSD1 dihydrochloride | 2102933-95-7 | 289.24 | 10mM | Histone Demethylase |
T3552 | CPI-455 | 1628208-23-0 | 278.32 | 10mM | Histone Demethylase |
T3719 | Daminozide | 1596-84-5 | 160.17 | 10mM | Histone Demethylase |
T4100 | AS8351 | 796-42-9 | 570.69 | 10mM | Histone Demethylase |
T4214 | KDM4D-IN-1 | 2098902-68-0 | 225.21 | 10mM | Histone Demethylase |
T4383 | GSK-J4 Hydrochloride | 1797983-09-5 | 453.97 | 10mM | Histone Demethylase |
T4418 | GSK2879552 2HCl (1401966-69-5(free base)) | T4418 | 437.41 | 10mM | Histone Demethylase |
T6073 | OG-L002 | 1357302-64-7 | 225.29 | 10mM | Histone Demethylase; HSV; monoamine oxidase |
T6545 | IOX1 | 5852-78-8 | 302.46 | 10mM | Histone Demethylase |
T6593 | ML324 | 1222800-79-4 | 349.43 | 10mM | Histone Demethylase; HSV |
T6847 | GSK-J1 | 1373422-53-7 | 389.45 | 10mM | Histone Demethylase |
T6922 | ORY1001 | 1431326-61-2 | 303.27 | 10mM | Histone Demethylase |
T4527 | Seclidemstat | 1423715-37-0 | 450.94 | 10mM | Histone Demethylase |
T5825 | Iadademstat dihydrochloride | 1431303-72-8 | 303.27 | 10mM | Histone Demethylase |
T7942 | Tranylcypromine hemisulfate | 13492-01-8 | 364.46 | 10mM | Histone Demethylase; MAO; monoamine oxidase |
T5484 | GSK467 | 1628332-52-4 | 319.32 | 10mM | Histone Demethylase; Histone Methyltransferase |
T13055 | T-3775440 hydrochloride | 1422535-52-1 | 346.85 | 10mM | Histone Demethylase |
T13748 | L-2-Hydroxyglutaric acid disodium | 63512-50-5 | 192.08 | 10mM | Histone Demethylase; Mitochondrial Metabolism |
TQ0050 | NCGC00244536 | 2003260-55-5 | 382.45 | 10mM | Histone Demethylase |
T15648 | KDM5-C70 | 1596348-32-1 | 336.43 | 10mM | Histone Demethylase |
T16435 | PBIT | 2514-30-9 | 241.31 | 10mM | Histone Demethylase; Histone Methyltransferase |
T11882 | Pulrodemstat benzenesulfonate | 2097523-60-7 | 609.64 | 10mM | Histone Demethylase |
T9243 | PFI-90 | 53995-62-3 | 214.22 | 10mM | Histone Demethylase |
T38318L | Acetyl Pentapeptide-1 acetate | T38318L | 721.8 | 10mM | Histone Demethylase |
T21652 | RN-1 dihydrochloride | 1781835-13-9 | 452.42 | 10mM | Histone Demethylase;MAO |
T15649 | KDM5-IN-1 | 1628210-26-3 | 324.38 | 10mM | Histone Demethylase |
T39989L | JQKD82 trihydrochloride | T39989L | 610.01 | 10mM | Histone Demethylase |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |