AMPK inhibitor/activator kit 包含AMP 依赖的蛋白激酶AMPK 抑制剂/激活剂,AMPK 是生物能量代谢调节的关键激酶,维持细胞生理活动的平稳运转,AMPK 能被机体各种刺激激活,包括细胞压力、运动、激素及能影响细胞代谢的物质,常用于研究肿瘤、衰老、糖尿病及其他代谢相关疾病。TargetMol 为您提供30种精选AMPK 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0800 | Danthron | 117-10-2 | 240.22 | 10mM | AMPK; Antibacterial; Autophagy; Virus Protease |
T1477 | AICAR | 2627-69-2 | 258.24 | 10mM | AMPK; Autophagy; Mitophagy; YAP |
T1977 | Dorsomorphin | 866405-64-3 | 399.49 | 10mM | AMPK; Autophagy; TGF-beta/Smad |
T2468 | A-769662 | 844499-71-4 | 360.39 | 10mM | AMPK; Fatty Acid Synthase |
T2854 | Phillyrin | 487-41-2 | 534.56 | 10mM | AMPK; Influenza Virus; P450 |
T3863 | Chikusetsusaponin IVa | 51415-02-2 | 794.98 | 10mM | AMPK |
T4427 | PF-06409577 | 1467057-23-3 | 341.79 | 10mM | AMPK |
T6146 | Dorsomorphin dihydrochloride | 1219168-18-9 | 472.41 | 10mM | AMPK; Autophagy; TGF-beta/Smad |
T6854 | GSK621 | 1346607-05-3 | 489.91 | 10mM | AMPK; Apoptosis; Autophagy |
T4S0800 | Demethyleneberberine | 25459-91-0 | 324.35 | 10mM | AMPK; HIF; NF-κB; NOS; P450 |
T5187 | MK-3903 | 1219737-12-8 | 454.9 | 10mM | AMPK |
T7362 | O-304 | 1261289-04-6 | 380.25 | 10mM | AMPK |
T7327 | 7-Methoxyisoflavone | 1621-56-3 | 252.26 | 10mM | AMPK |
T8476 | RSVA405 | 140405-36-3 | 312.37 | 10mM | AMPK; Autophagy; STAT |
T8432 | ASP4132 | 1640294-30-9 | 937.06 | 10mM | AMPK |
T8526 | Metformin | 657-24-9 | 129.16 | 10mM | AMPK; Autophagy; Mitophagy |
T16156 | MT 63-78 | 1179347-65-9 | 326.35 | 10mM | AMPK; Apoptosis; mTOR |
T16099 | MK8722 | 1394371-71-1 | 449.89 | 10mM | AMPK |
T13265 | Urolithin B | 1139-83-9 | 212.2 | 10mM | Akt; AMPK; Endogenous Metabolite; ERK; JNK; NF-κB |
T8740 | COH-SR4 | 73439-19-7 | 350.02 | 10mM | AMPK |
TQ0028 | EX229 | 1219739-36-2 | 431.87 | 10mM | AMPK |
T2S0820 | Karanjin | 521-88-0 | 292.29 | 10mM | AMPK; Apoptosis |
T8929 | BC1618 | 2222094-18-8 | 415.45 | 10mM | AMPK; E1/E2/E3 Enzyme; Mitophagy |
TN1499 | Cimiracemoside C | 256925-92-5 | 620.8 | 10mM | AMPK |
TN6751 | 1-HEXACOSANOL | 506-52-5 | 382.71 | 10mM | AMPK; NPC1L1 |
T20029 | Buformin hydrochloride | 1190-53-0 | 193.68 | 10mM | AMPK |
T19661 | 8-Chloroadenosine | 34408-14-5 | 301.69 | 10mM | AMPK |
T13411 | ZLN024 | 723249-01-2 | 325.22 | 10mM | AMPK |
T41162 | ZLN 024 hydrochloride | 1883548-91-1 | 361.68 | 10mM | AMPK |
T24626 | PF-249 | 1467059-70-6 | 345.78 | 10mM | AMPK |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |