Akt inhibitor/activator kit 包含蛋白激酶Akt 抑制剂/激活剂,Akt 是经典的PI3K-AKT-mTOR 信号通路的中心环节,调节肿瘤细胞生长、增殖、促进细胞侵袭和转移、促进新生血管生成,还使肿瘤细胞产生化疗、放疗耐受性。TargetMol 为您提供37种精选Akt 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1920 | Capivasertib | 1143532-39-1 | 428.92 | 10mM | Akt; Autophagy; mTOR; PKA |
T1952 | MK-2206 dihydrochloride | 1032350-13-2 | 480.39 | 10mM | Akt; Apoptosis; Autophagy |
T2274 | SC79 | 305834-79-1 | 364.78 | 10mM | Akt |
T2420 | PHT-427 | 1191951-57-1 | 409.61 | 10mM | Akt; Apoptosis; PDK |
T2482 | AT13148 | 1056901-62-2 | 313.78 | 10mM | Akt; PKA; ROCK; S6 Kinase; SGK |
T2492 | Perifosine | 157716-52-4 | 461.66 | 10mM | Akt; Apoptosis; Autophagy |
T2790 | Oridonin | 28957-04-2 | 364.44 | 10mM | Akt; Antibacterial |
T3132 | SC66 | 871361-88-5 | 276.33 | 10mM | Akt; Apoptosis |
T3346 | AKT inhibitor VIII | 612847-09-3 | 551.64 | 10mM | Akt; Apoptosis |
T3467 | Miransertib | 1313881-70-7 | 432.53 | 10mM | Akt; Parasite |
T3861 | Isobavachalcone | 20784-50-3 | 324.38 | 10mM | Akt; Apoptosis; Autophagy; Reactive Oxygen Species |
T6065 | Triciribine | 35943-35-2 | 320.3 | 10mM | Akt; DNA/RNA Synthesis; HIV Protease |
T6252 | Ipatasertib | 1001264-89-6 | 458 | 10mM | Akt |
T6285 | GSK-690693 | 937174-76-0 | 425.48 | 10mM | Akt; AMPK; Autophagy; PKC; Serine Protease |
T6304 | AT7867 | 857531-00-1 | 337.85 | 10mM | Akt; PKA; S6 Kinase |
T6817 | Deguelin | 522-17-8 | 394.42 | 10mM | Akt; Apoptosis; Autophagy; PI3K |
T6849 | Uprosertib | 1047634-65-0 | 429.25 | 10mM | Akt |
T4489 | AKT-IN-1 | 1357158-81-6 | 343.42 | 10mM | Akt |
T5S0896 | Loureirin A | 119425-89-7 | 286.32 | 10mM | Akt; PI3K |
T7315 | BAY1125976 | 1402608-02-9 | 383.45 | 10mM | Akt |
T7885 | Afuresertib hydrochloride | 1047645-82-8 | 463.8 | 10mM | Akt; PKC; ROCK |
T7879 | TASP0415914 | 1292300-75-4 | 323.37 | 10mM | Akt; PI3K |
T5508 | PF-AKT400 | 1004990-28-6 | 400.43 | 10mM | Akt |
T6S0619 | Pachymic acid | 29070-92-6 | 528.77 | 10mM | Akt; ERK |
T16104 | ML-9 | 105637-50-1 | 361.29 | 10mM | Akt; Myosin |
T6139L | A-674563 2HCl(552325-73-2(fb-2hcl)) | T6139L | 431.36 | 10mM | Akt; CDK; ERK; PKA; PKC |
T8969 | API-1 | 36707-00-3 | 337.29 | 10mM | Akt |
T8427 | Borussertib | 1800070-77-2 | 596.68 | 10mM | Akt |
T14034 | 3CAI | 28755-03-5 | 193.63 | 10mM | Akt |
T9393 | (E)-Akt inhibitor-IV | 959841-49-7 | 616.56 | 10mM | Akt |
T14072 | A-443654 | 552325-16-3 | 397.47 | 10mM | Akt; Casein Kinase; CDK; Chk; ERK; FLT; GSK-3; MAPK; PKA; PKC; S6 Kinase; Src; VEGFR |
T13376 | YS-49 | 132836-42-1 | 386.28 | 10mM | Adrenergic Receptor; Akt; PI3K; RAAS |
T25150 | BI-69A11 | 1233322-09-2 | 425.87 | 10mM | Akt; NF-κB |
T6303L | CCT128930 hydrochloride | 2453324-32-6 | 378.3 | 10mM | Akt; Apoptosis; Autophagy; mTOR; PKA |
T15374 | Ipatasertib dihydrochloride | 1396257-94-5 | 530.92 | 10mM | Akt; PKA |
T23695 | Akt-I-1,2 | 473382-50-2 | 375.89 | 10mM | Akt |
T25017 | AKT-I-1 | 473382-39-7 | 378.51 | 10mM | Akt |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |