AChR antagonist/agonist kit 包含乙酰胆碱受体AChR 拮抗剂/激动剂,AChR 主要包括烟碱型和毒蕈碱型受体,毒蕈碱型受体产生副交感神经兴奋效应,抑制心脏活动,收缩支气管胃肠平滑肌和膀胱逼尿肌,增加消化腺分泌,缩小瞳孔等。烟碱型受体引起自主神经节的节后神经元兴奋,导致骨骼肌兴奋。TargetMol 为您提供131种精选AChR 拮抗剂/激动剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0072 | Adiphenine hydrochloride | 50-42-0 | 347.88 | 10mM | AChR |
T0099 | Tolterodine tartrate | 124937-52-6 | 475.58 | 10mM | AChR |
T0166 | Pancuronium dibromide | 15500-66-0 | 732.67 | 10mM | AChR |
T0177 | Homatropine Bromide | 51-56-9 | 356.26 | 10mM | AChR |
T0253 | Methscopolamine | 155-41-9 | 398.29 | 10mM | AChR |
T0268 | Lobeline hydrochloride | 134-63-4 | 373.92 | 10mM | AChR |
T0287 | Hexamethonium Bromide | 55-97-0 | 362.19 | 10mM | AChR; Apoptosis; Dopamine Receptor |
T0333 | Aniracetam | 72432-10-1 | 219.24 | 10mM | 5-HT Receptor; AChR; Dopamine Receptor; GluR; iGluR |
T0703 | Flavoxate hydrochloride | 3717-88-2 | 427.92 | 10mM | AChR |
T0786 | Clidinium bromide | 3485-62-9 | 432.35 | 10mM | AChR |
T0804 | Pilocarpine Hydrochloride | 54-71-7 | 244.72 | 10mM | AChR |
T0818 | Decamethonium bromide | 541-22-0 | 418.29 | 10mM | AChE; AChR |
T0862 | Diphenidol hydrochloride | 3254-89-5 | 345.91 | 10mM | AChR; Sodium Channel |
T0962 | L-Hyoscyamine | 101-31-5 | 289.38 | 10mM | AChR |
T1006 | Propantheline bromide | 50-34-0 | 448.4 | 10mM | AChR |
T1039 | Choline chloride | 67-48-1 | 139.63 | 10mM | AChR |
T1049 | Oxybutynin chloride | 1508-65-2 | 393.96 | 10mM | AChR; Potassium Channel |
T1179 | Tiotropium bromide | 136310-93-5 | 472.42 | 10mM | AChR |
T1221 | Acetylcholine chloride | 60-31-1 | 181.66 | 10mM | AChR; Calcium Channel; Endogenous Metabolite |
T1281 | Tropicamide | 1508-75-4 | 284.36 | 10mM | AChR |
T1285 | Anethole trithione | 532-11-6 | 240.35 | 10mM | AChR |
T1328 | DL-trihexyphenidyl hydrochloride | 58947-95-8 | 337.93 | 10mM | AChR |
T1341 | Nortropine | 538-09-0 | 127.18 | 10mM | AChR |
T1460 | Dicyclomine hydrochloride | 67-92-5 | 345.95 | 10mM | AChR |
T1472 | Trospium chloride | 10405-02-4 | 427.97 | 10mM | AChR |
T1474 | Otilonium bromide | 26095-59-0 | 563.57 | 10mM | AChR; Calcium Channel |
T1534 | Darifenacin hydrobromide | 133099-07-7 | 505.45 | 10mM | AChR |
T1542 | Pirenzepine dihydrochloride | 29868-97-1 | 424.32 | 10mM | AChR |
T1657 | Varenicline Tartrate | 375815-87-5 | 361.35 | 10mM | AChR |
T1682 | Methacholine Chloride | 62-51-1 | 195.69 | 10mM | AChR |
T1760 | TBPB | 634616-95-8 | 404.55 | 10mM | AChR |
T2138 | Oxyphencyclimine Hydrochloride | 125-52-0 | 380.91 | 10mM | AChR |
T2141 | Mecamylamine hydrochloride | 826-39-1 | 203.75 | 10mM | AChR |
T2182 | Scopolamine hydrobromide trihydrate | 6533-68-2 | 438.31 | 10mM | AChR |
T2183 | Scopolamine butylbromide | 149-64-4 | 440.37 | 10mM | AChR |
T2198 | Arecoline hydrobromide | 300-08-3 | 236.11 | 10mM | AChR |
T2285 | Encenicline hydrochloride | 550999-74-1 | 357.3 | 10mM | AChR |
T2387 | Glycopyrrolate | 596-51-0 | 398.33 | 10mM | AChR |
T2422 | PNU-282987 | 123464-89-1 | 301.21 | 10mM | AChR |
T2555 | Aclidinium bromide | 320345-99-1 | 564.55 | 10mM | AChR |
T2663 | GTS-21 dihydrochloride | 156223-05-1 | 381.3 | 10mM | 5-HT Receptor; AChR |
T3126 | Bethanechol chloride | 590-63-6 | 196.68 | 10mM | AChR |
T3619 | VU0357017 hydrochloride | 1135242-13-5 | 369.89 | 10mM | AChR |
T6364 | Desfesoterodine | 207679-81-0 | 341.49 | 10mM | AChR |
T6547 | Ipratropium Bromide | 22254-24-6 | 412.37 | 10mM | AChR |
T6548 | Irsogladine | 57381-26-7 | 256.09 | 10mM | AChR; PDE |
T6575 | LY2119620 | 886047-22-9 | 437.94 | 10mM | AChR |
T6607 | Nitenpyram | 150824-47-8 | 270.72 | 10mM | AChR |
T6684 | Succinylcholine Chloride Dihydrate | 6101-15-1 | 397.34 | 10mM | AChR |
T6744 | Methylbenactyzium Bromide | 3166-62-9 | 422.36 | 10mM | AChR |
T6950 | PNU-120596 | 501925-31-1 | 311.72 | 10mM | AChR |
T7002 | Trihexyphenidyl hydrochloride | 52-49-3 | 337.93 | 10mM | AChR |
T4S1619 | L-Hyoscyamine sulfate | 620-61-1 | 676.8 | 10mM | AChR |
T5S0106 | Peimisine | 19773-24-1 | 427.62 | 10mM | AChR; RAAS |
T3865 | beta-Eudesmol | 473-15-4 | 222.37 | 10mM | AChR; TRP/TRPV Channel |
T7079 | Batefenterol | 743461-65-6 | 740.24 | 10mM | AChR; Adrenergic Receptor |
T4986 | Imidafenacin | 170105-16-5 | 319.4 | 10mM | AChR |
T4997 | Umeclidinium bromide | 869113-09-7 | 508.49 | 10mM | AChR |
T5051 | Isopropamide Iodide | 71-81-8 | 480.43 | 10mM | AChR |
T7124 | Dinotefuran | 165252-70-0 | 202.21 | 10mM | AChR; Parasite |
T5805 | Guvacoline hydrochloride | 6197-39-3 | 177.63 | 10mM | AChR |
T7193 | Encenicline | 550999-75-2 | 320.84 | 10mM | AChR |
T7392 | Revefenacin | 864750-70-9 | 597.75 | 10mM | AChR |
T7422 | CCMI | 917837-54-8 | 388.25 | 10mM | AChR |
T7561 | Benzetimide hydrochloride | 5633-14-7 | 398.93 | 10mM | AChR |
T7405 | Piperidolate | 82-98-4 | 323.43 | 10mM | AChR |
T7780 | Blarcamesine | 195615-83-9 | 281.39 | 10mM | AChR |
T7884 | NS 1738 | 501684-93-1 | 365.14 | 10mM | AChR |
T7895 | Syn-Ake acetate | 823202-99-9 | 495.58 | 10mM | AChR |
T8007 | VU 0238429 | 1160247-92-6 | 351.28 | 10mM | AChR |
T8383 | Cyclopentolate Hydrochloride | 5870-29-1 | 327.85 | 10mM | AChR |
T8224 | VU0119498 | 79183-37-2 | 316.15 | 10mM | AChR |
T8219 | VU0238441 | 85511-68-8 | 339.7 | 10mM | AChR |
T8318 | BNC210 | 13589-06-5 | 317.38 | 10mM | AChR |
T14094 | Acetamiprid | 135410-20-7 | 222.67 | 10mM | AChR |
T8725 | A 582941 HCl (848591-90-2(free base)) | T8725 | 316.83 | 10mM | AChR |
T13066 | TAK-071 | 1820812-16-5 | 421.46 | 10mM | AChR |
T8868 | 4BP-TQS | 360791-49-7 | 405.31 | 10mM | AChR |
TQ0117 | A-867744 | 1000279-69-5 | 402.89 | 10mM | AChR; Autophagy |
T15942 | MK-7622 | 1227923-29-6 | 399.48 | 10mM | AChR |
T21153 | Clothianidin | 210880-92-5 | 249.67 | 10mM | AChR |
T23348 | SEN12333 | 874450-44-9 | 339.43 | 10mM | AChR |
T12165 | nAChR agonist 1 | 1394371-75-5 | 419.95 | 10mM | AChR |
T17300 | (-)-(S)-B-973B | 2244989-34-0 | 452.5 | 10mM | AChR |
T28827 | Sofpironium bromide | 1628106-94-4 | 470.4 | 10mM | AChR |
T23524 | W-84 dibromide | 21093-51-6 | 708.52 | 10mM | AChR |
T12489 | Pimethixene | 314-03-4 | 293.43 | 10mM | 5-HT Receptor; AChR; Dopamine Receptor; Histamine Receptor |
T28069 | ML380 | 1627138-52-6 | 494.53 | 10mM | AChR |
T23469 | TQS | 353483-92-8 | 376.47 | 10mM | AChR |
T23146 | PHA 568487 free base | 527680-56-4 | 288.34 | 10mM | AChR |
T8147 | Solifenacin | 242478-37-1 | 362.46 | 10mM | AChR |
T12201 | Nebracetam hydrochloride | 1177279-49-0 | 240.73 | 10mM | AChR |
T14345 | Atropine methyl bromide | 2870-71-5 | 384.31 | 10mM | AChR |
T11095L | DREADD agonist 21 | 56296-18-5 | 278.35 | 10mM | 5-HT Receptor; AChR; Adrenergic Receptor; Histamine Receptor |
T17238 | VU0152100 | 409351-28-6 | 341.43 | 10mM | AChR |
T23513 | VU10010 | 633283-39-3 | 345.85 | 10mM | AChR |
T29123 | VU0152099 | 612514-42-8 | 355.41 | 10mM | AChR |
T9419 | Fesoterodine | 286930-02-7 | 411.58 | 10mM | AChR |
T9353 | OXOMEMAZINE | 3689-50-7 | 330.44 | 10mM | AChR; Histamine Receptor |
T22735 | DMAB-anabaseine dihydrochloride | 154149-38-9 | 364.31 | 10mM | AChR |
T22448 | Tropisetron | 89565-68-4 | 284.35 | 10mM | 5-HT Receptor; AChR |
T13325 | VU 0365114 | 1208222-39-2 | 397.35 | 10mM | AChR |
T17244 | VU0467154 | 1451993-15-9 | 444.45 | 10mM | AChR |
T23116 | Oxotremorine sesquifumarate | 17360-35-9 | 380.4 | 10mM | AChR |
T23071 | Nitrocaramiphen hydrochloride | 98636-73-8 | 370.87 | 10mM | AChR |
T9542 | NS3861 | 216853-59-7 | 284.21 | 10mM | AChR |
T28199 | NS9283 | 913830-15-6 | 248.24 | 10mM | AChR |
T29137 | VU0453595 | 1432436-13-9 | 322.34 | 10mM | AChR |
T28531 | Facinicline hydrochloride | 677305-02-1 | 306.79 | 10mM | 5-HT Receptor; AChR |
T13385 | Zamifenacin fumarate | 127308-98-9 | 531.6 | 10mM | AChR |
T38272 | Thiacloprid | 111988-49-9 | 252.72 | 10mM | AChR; Parasite |
T9787 | suvn-911 | 2414674-71-6 | 224.69 | 10mM | AChR |
T23508 | VU 0255035 | 1135243-19-4 | 432.52 | 10mM | AChR |
T16563L | Pozanicline hydrochloride | T16563L | 228.72 | 10mM | AChR |
T19940 | Sulfoxaflor | 946578-00-3 | 276.26 | 10mM | AChR |
T37196 | 5-AAM-2-CP | 175424-74-5 | 184.62 | 10mM | AChR |
T9694 | Emraclidine | 2170722-84-4 | 390.4 | 10mM | AChR |
T9889 | M4 mAChR agonist-1 | 785705-53-5 | 290.38 | 10mM | AChR |
T9877 | tiquizium | 149755-23-7 | 330.53 | 10mM | AChR |
T16411 | Otenzepad | 102394-31-0 | 421.54 | 10mM | AChR |
T60080 | TMPH | 849461-90-1 | 269.42 | 10mM | AChR |
TN1519L | (-)-Coclaurine hydrochloride | 3422-42-2 | 321.8 | 10mM | AChR |
T23286 | S 24795 | 304679-75-2 | 418.07 | 10mM | AChR |
T14333 | Asoxime dichloride | 34433-31-3 | 359.21 | 10mM | AChR |
T19870 | Aceclidine | 827-61-2 | 169.22 | 10mM | AChR |
T12339 | Oxotremorine M iodide | 3854-04-4 | 322.19 | 10mM | AChR |
T10108 | 3-Bromocytisine | 207390-14-5 | 269.14 | 10mM | AChR |
T37818 | bPiDDB | 525596-66-1 | 514.38 | 10mM | AChR |
T12820 | S16961 | 153874-14-7 | 674.01 | 10mM | AChR |
T11588 | Hydroxybupropion | 92264-81-8 | 255.74 | 10mM | Norepinephrine;AChR |
T25538 | Iperoxo | 247079-84-1 | 324.16 | 10mM | AChR |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |