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Cat. No. | Product Name | Target | Signaling Pathways |
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T1305 |
Ceftazidime
GR20263,头孢他啶 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ceftazidime (GR20263) 是可静脉内或肌肉给药的第头孢菌素。它对革兰氏阳性和革兰氏阴性需氧细菌有体外活性。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。 | |||
T37465 |
CAY10742
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CAY10742 is an orally bioavailable oxadiazole antibiotic.1It is active against the Gram-positive bacteriaS. aureus,S. epidermidis,S. haemolyticus,B. cereus,B. licheniformis,E. faecalis, andE. faecium(MICs = 1-4 μg/ml), including laboratory strains and clinical isolates with varying degrees of resistance to methicillin, vancomycin, linezolid, and other antibiotics. CAY10742 (40 mg/kg) reduces the number of bacteria in mouse neutropenic thigh models of linezolid-sensitive or -resistant methicillin... | |||
T79735 |
DHFR-IN-9
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DHFR-IN-9(化合物8A)是一种二氢叶酸还原酶(DHFR)抑制剂,通过干扰细胞内嘌呤和胸苷酸的生物合成而影响细胞生长和增殖。该化合物对抗耐甲氧西林金黄色葡萄球菌(MRSA)ATCC 43300展现出显著的抑制效果(IC50=0.25 μg/mL),并在全身及大腿感染的小鼠模型中显示出抗感染能力(剂量:2.5 mg/kg,5 mg/kg;ip)。此外,DHFR-IN-9在乳腺癌小鼠模型中展示了超过紫杉醇(Y-B0015)的抗癌活性(剂量:2.5 mg/kg;ip;每3天1次)。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T8261 |
Ceftazidime Pentahydrate
头孢他啶五水合物,头孢他啶 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ceftazidime pentahydrate 是一种β-内酰胺类抗菌剂,对革兰氏阳性和革兰氏阴性需氧细菌有广谱活性,可静脉内或肌肉给药。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。 |