Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20237 |
Fenhexamid
Elevate,Teldor,环酰菌胺 |
Antifungal | Microbiology/Virology |
Fenhexamid (Elevate) 是一种甾醇生物合成抑制剂,对植物病原真菌具有抗真菌活性。 Fenhexamid 用于农业,并在水果和蔬菜中以可测量的量存在。 | |||
T20691 |
Fenpropidin
苯锈啶,Ro12-3049,Ro-12-3049,Ro 12-3049 |
Antifungal | Microbiology/Virology |
Fenpropidin (Ro-12-3049) 是甾醇类生物合成的抑制剂,具有杀菌的活性。 | |||
T14362 |
AY 9944
|
Others | Others |
AY 9944 是特异性的胆固醇生物合成抑制剂。它抑制 7- 脱氢胆固醇 Δ7- 还原酶 (IC50:13 nM),导致胆固醇不足和 7DHC 积累。在高剂量下,它可在培养的胚胎中抑制固醇 Δ7-Δ8 异构酶,造成胆固醇 8-en-3β-ol 的积累。 | |||
T68219 |
Peraclopone
|
||
Peraclopone is a hypolidemic drug. It is an inhibitor of 7-Dehydrocholesterol reductase. Peraclopone potently inhibits the final step in cholesterol biosynthesis. Feeding this agent to rats leads to a rapid replacement of membrane cholesterol with its immediate precursor 7-dehydrocholesterol, and a dramatic reduction in plasma sterol concentration. Peraclopone caused a dose-dependent decrease in cholesterol and a concomitant accumulation of provitamin D3 (7-dehydrocholesterol) in the skin, which... |