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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T67988 Embeconazole

R 120758,CS 758

Antifungal Microbiology/Virology
Embeconazole (R 120758) 是一种三唑类抗真菌剂。Embeconazole 对念珠菌、曲霉菌、新型隐球菌等临床重要真菌具有较强的体外活性。
T23955 Dactylfungin B

Dactylfungins B is a novel antifungal antibiotic produced by Dactylaria Parvispora. The antibiotics were active against Candida pseudotropicalis and other fungi, with a MIC value of fewer than 10 micrograms/ml.
T23954 Dactylfungin A

Dactylfungins A is a novel antifungal antibiotic produced by Dactylaria Parvispora. The antibiotics were active against Candida pseudotropicalis and other fungi, with a MIC value of fewer than 10 micrograms/ml.
T75176 Antifungal agent 53

Antifungal agent 53 (A03) 是一种有效的白色念珠菌 CYP51抑制剂,具有抗真菌活性。Antifungal agent 53 阻止真菌生物膜的形成。Antifungal agent 53 也显示出良好的安全性。
T68562 FTR-1335

FTR1335 is a CaNMT inhibitor (IC50 = 0.49 nM) with good fungal selectivity. CaNMT inhibitors are fungicidal and show antifungal activity against Candida (especially fluconazole-resistant strains). They function by inhibiting N-myristoyltransferase (NMT), which catalyzes the transfer of a C14 fatty acif from myristoyl-CoA to the N-terminal of glycine in many fungal proteins. Without this process, fungi can die. This process also occurs in humans, and as such selectivity is an important characteri...
T79413 Antifungal agent 73

Antifungalagent 73 (compound A32)是一款用于治疗唑类耐药Candida感染的抗真菌药物。该化合物通过破坏真菌的细胞壁和细胞膜来发挥作用,并且针对病原真菌和氟康唑(Fluconazole)耐药菌株显示出有效的体内抗真菌活性。
T21881 Fluconazole hydrate

Fluconazole 水合物是抗真菌化合物,用于治疗和预防浅表和全身性的真菌感染。

化合物

Embeconazole
Cat.No: T67988
Synonym: R 120758,CS 758
Target: Antifungal
Dactylfungin B
Cat.No: T23955
Synonym:
Target:
Dactylfungin A
Cat.No: T23954
Synonym:
Target:
Antifungal agent 53
Cat.No: T75176
Synonym:
Target:
FTR-1335
Cat.No: T68562
Synonym:
Target:
Antifungal agent 73
Cat.No: T79413
Synonym:
Target:
Fluconazole hydrate
Cat.No: T21881
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1388 Fluconazole

氟康唑,UK-49858

Antibiotic; Antifection; Antifungal Microbiology/Virology
Fluconazole (UK-49858) 是一种对多种真菌具有活性的三唑类抗真菌剂,抑制 C. albicans 和 Candida kefyr 的 IC99为 0.20 μg/mL 至 0.39 μg/mL。

天然产物

Fluconazole
Cat.No: T1388
Synonym: 氟康唑,UK-49858
Target: Antibiotic, Antifection, Antifungal
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