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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T4989 Fosfomycin Tromethamine

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T3131 Fosfomycin calcium

Phosphomycin calcium salt,Fosmicin,磷霉素钙

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T77254 Maltodextrin, dextrose equivalent 16.5-19.5

Maltodextrin(麦芽糊精),dextrose equivalent(葡萄糖当量)为16.5-19.5,可作为药用辅料。药用辅料,亦称药用助剂,非药物成分的化学物质,用于辅助药物制剂过程。此类辅料提升药物制剂的稳定性、溶解性及加工性,同时影响药物的吸收、分布、代谢及排泄(ADME)过程。
T68765 Spirorenone

Spirorenone is an androstadienone derivative as a highly effective aldosterone antagonist. Spirorenone is 8.6 times as potent as spironolactone, but showed a lower affinity for the mineralocorticoid receptors. In phase I clinical trials Spirorenone was absorbed with a half-life of 20-30 min, achieving maximum concentrations of about 100 ng/ml (10 mg) and 260 ng/ml (40 mg) after 1-2 h. Disposition of the parent drug was biphasic with half-lives of 50-60 min (distribution) and 5-6 h (elimination)....
T77228 Polyoxyethylene Sorbitan Monostearate

Polyoxyethylene Sorbitan Monostearate 是一种由饱和脂肪酸硬脂酸 (C18:0) 构成的酯,广泛应用作药用辅料,包括表面活性剂、乳化剂、增溶剂和润湿剂。作为药用助剂,其主要作用是改善药物制剂的稳定性、溶解性和加工性,同时对药物的吸收、分布、代谢和消除 (ADME) 过程具有影响。
T73620 Poly(acrylic acid)

Poly(acrylic acid) 通过吸附作用在金属表面形成保护层,有效抑制纯铸铝在酸性介质中的腐蚀现象。此外,Poly(acrylic acid) 还可作为药物制剂中的包衣材料、释放阻断剂等药用辅料使用。药用辅料,亦称药用助剂,是指在制药过程中,除药物活性成分外使用的其他化学物质。这些辅料通常作为非活性成分加入药物制剂中,旨在提升制剂的稳定性、溶解性及加工性。同时,药用辅料对药物的吸收、分布、代谢与排泄(ADME)过程也具有一定影响。
T37800 PF-04449613

PF-04449613 is a phosphodiesterase 9A (PDE9A) inhibitor (IC50= 22 nM).1It is selective for PDE9A over PDE1C (IC50= >1,000 nM), as well as over a variety of other PDEs, inhibiting PDE2-8, -10, and -11 activity by less than 30% in a panel of enzymes, ion channels, and transporters at 1 μM but does inhibit the human dopamine transporter (DAT; Ki= 293 nM). PF-04449613 (0.1-100 mg/kg, s.c.) increases cerebrospinal fluid (CSF) levels of cyclic GMP (cGMP) in rats. Subcutaneous administration of PF-0444...

化合物

Fosfomycin Tromethamine
Cat.No: T4989
Synonym:
Target: Antibacterial, Antibiotic
Fosfomycin calcium
Cat.No: T3131
Synonym: Phosphomycin calcium salt,Fosmicin,磷霉素钙
Target: Antibacterial, Antibiotic
Maltodextrin, dextrose equivalent 16.5-19.5
Cat.No: T77254
Synonym:
Target:
Spirorenone
Cat.No: T68765
Synonym:
Target:
Polyoxyethylene Sorbitan Monostearate
Cat.No: T77228
Synonym:
Target:
Poly(acrylic acid)
Cat.No: T73620
Synonym:
Target:
PF-04449613
Cat.No: T37800
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。

天然产物

Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
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