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7

抑制剂 & 化合物

3

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T71714 hClpP-activator-D9

hClpP-activator-D9 is a novel potent and species-selective activator of human ClpP (hClpP).
T70842 ACP1b

ACP1b is an activator of ClpP protease.
T73314 (R)-ZG197

(R)-ZG197为一种对金黄色葡萄球菌酪蛋白溶解蛋白酶P (SaClpP) 具有高选择性的激活剂,EC50值为1.5 μM。此外,(R)-ZG197还能激活人类ClpP (HsClpP),其EC50为31.4 μM。
T10125 (3R,4R)-A2-32-01

Others Others
(3R,4R)-A2-32-01 (compound 2) is a specific caseinolytic protein proteases (ClpP) inhibitor (EC50: 4.5 μM).
T72657 (3S,4S)-A2-32-01

(3S,4S)-A2-32-01 ,A2-32-01 的活性较低的 (S,S)-对映异构体。A2-32-01 是一种有效的酪蛋白分解蛋白蛋白酶 (ClpP) 抑制剂。
T73315 (S)-ZG197

(S)-ZG197为高选择性金黄色葡萄球菌酪蛋白溶解蛋白酶P (SaClpP) 激活剂,EC50值为1.4μM。
T80737 ZG36

ZG36是一种人类Caseinolytic protease P(ClpP)激动剂,具有非选择性地降解呼吸链复合物和减少线粒体DNA的能力,从而导致线粒体功能衰竭及白血病细胞死亡。此外,ZG36能够抑制异种移植小鼠模型中急性髓细胞性白血病的发展。

化合物

hClpP-activator-D9
Cat.No: T71714
Synonym:
Target:
ACP1b
Cat.No: T70842
Synonym:
Target:
(R)-ZG197
Cat.No: T73314
Synonym:
Target:
(3R,4R)-A2-32-01
Cat.No: T10125
Synonym:
Target: Others
(3S,4S)-A2-32-01
Cat.No: T72657
Synonym:
Target:
(S)-ZG197
Cat.No: T73315
Synonym:
Target:
ZG36
Cat.No: T80737
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-00408 ClpP Protein, Clostridium botulinum, Recombinant (His & SUMO)

clpP,Endopeptidase Clp,ATP-dependent Clp protease p...

Clostridium botulinum E. coli
ClpP Protein, Clostridium botulinum, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-00209 CLPP2 Protein, Borrelia burgdorferi, Recombinant (His & Myc)

clpP-2,Endopeptidase Clp 2,ATP-dependent Clp protea...

Borrelia burgdorferi E. coli
Cleaves peptides in various proteins in a process that requires ATP hydrolysis. Has a chymotrypsin-like activity. Plays a major role in the degradation of misfolded proteins.
TMPH-00582 Endopeptidase Clp Protein, E. coli, Recombinant (His & Myc)

clpP,ATP-dependent Clp protease proteolytic subunit...

E. coli E. coli
Cleaves peptides in various proteins in a process that requires ATP hydrolysis. Has a chymotrypsin-like activity. Plays a major role in the degradation of misfolded proteins.

重组蛋白

ClpP Protein, Clostridium botulinum, Recombinant (His & SUMO)
Cat.No: TMPH-00408
Species: Clostridium botulinum
Expression System: E. coli
CLPP2 Protein, Borrelia burgdorferi, Recombinant (His & Myc)
Cat.No: TMPH-00209
Species: Borrelia burgdorferi
Expression System: E. coli
Endopeptidase Clp Protein, E. coli, Recombinant (His & Myc)
Cat.No: TMPH-00582
Species: E. coli
Expression System: E. coli
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