Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3710 |
XMD16-5
|
Tyrosinase; PPAR | DNA Damage/DNA Repair; Metabolism; Proteases/Proteasome |
XMD16-5 是TNK2抑制剂,对D163E 和R806Q 突变体的IC50值分别为16和77nM。 | |||
T3709 |
XMD8-87
ACK1-B19 |
Tyrosinase; PPAR | DNA Damage/DNA Repair; Metabolism; Proteases/Proteasome |
XMD8-87 (ACK1-B19)是TNK2抑制剂,对于D163E 和R806Q 突变体的IC50值分别为38和113 nM。 |