Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13077 |
Taniborbactam dihydrochloride
VNRX-5133 dihydrochloride,Taniborbactam 2HCl |
Antibacterial; Antifungal | Microbiology/Virology |
Taniborbactam dihydrochloride (VNRX-5133 dihydrochloride) 是一种具有选择性和有效性的新型环硼酸β-内酰胺酶抑制剂,具有抗菌活性,对革兰氏阴性菌抑制作用显著。Taniborbactam dihydrochloride 抑制 KPC-2,AmpC,OXA-48 和 VIM-2 ,可以用于研究真菌感染。 | |||
T24942 |
VNRX-5133
VNRX 5133 |
||
VNRX-5133 is an injectable broad-spectrum β-lactamase inhibitor. VNRX-5133 is a novel β-lactamase inhibitor with potent and selective direct inhibitory activity against both serines- and Metallo-β-lactamases. | |||
T13077L |
Taniborbactam
VNRX-5133 |
Antibacterial | Microbiology/Virology |
Taniborbactam is a reversible and selective boronic acid-containing pan-spectrum β-lactamase inhibitor (IC50s: 8-530 nM). Taniborbactam has IC50s of 30 nM, 32 nM, 42 nM, 20 nM for KPC-2, AmpC, OXA-48, and VIM-2. |