Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79401 |
Tyrosinase-IN-13
|
Tyrosinase | Proteases/Proteasome |
Tyrosinase-IN-13 (compound 3c)为Flurbiprofen的衍生物,具有非竞争性酪氨酸酶抑制活性(IC50=68 μM;Ki=36.3 μM),并对肝细胞癌(HepG2)、结直肠癌(HT-29)及黑色素瘤(B16F10)细胞表现出细胞毒性。 |