Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13133 |
Tetrabenazine Metabolite
(-)-β-Dihydrotetrabenazine,(-)-β-HTBZ |
Monoamine Transporter | Membrane transporter/Ion channel |
Tetrabenazine Metabolite ((-)-β-HTBZ) 是一种囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,是 Tetrabenazine 的一种活性代谢物。Tetrabenazine Metabolite 对 VMAT2 具有高亲和力,其Ki 为13.4 nM。Tetrabenazine Metabolite 常常被用于研究与亨廷顿氏病和其他多动障碍相关的舞蹈病。 | |||
T23983 |
Deutetrabenazine metabolite M4
SD-1018,Deuterated monohydroxy tetrabenazine,D6-tetrabenazine metabolite M4 |
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Deutetrabenazine metabolite M4 is believed to be related to its effect as a reversible depletion of monoamines from nerve terminals. The major circulating metabolites of Deutetrabenazine, are reversible inhibitors of VMAT2, resulting in decreased uptake | |||
T12190 |
Trans (2,3)-Dihydrotetrabenazine
(2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine |
Others | Others |
Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2). |