Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T75240 | Taltobulin hydrochloride | ||
Taltobulin hydrochloride (HTI-286 hydrochloride) 是一种合成的三肽半胱氨酸类似物,为高效抗微管剂,能够在体内外绕过P-糖蛋白介导的药物耐药性。该化合物通过抑制微管蛋白的聚合和破坏细胞内微管结构,进而引起细胞有丝分裂停滞和细胞凋亡。 | |||
T13073L |
Taltobulin hydrochloride (228266-40-8 free base)
SPA-110 hydrochloride,Taltobulin hydrochloride,HTI-286 hydrochloride |
Others | Others |
Taltobulin hydrochloride is a synthetic analogue of the tripeptide hemiasterlin, is a potent agent of antimicrotubule that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. |