Cat. No. | Product Name | Target | Signaling Pathways |
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T79054 |
TRPC3/6-IN-2
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TRPC3/6-IN-2为针对TRPC3及TRPC6的高效抑制剂,IC50分别为16 nM对TRPC3与29.8 nM对TRPC6。 | |||
T71303 |
Flufenamic Acid-d4
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Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear... |