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Cat. No. Product Name Target Signaling Pathways
TP2021 [Pro3]-GIP (Rat)

High affinity rat GIP receptor partial agonist (Kd = 13 nM). Increases cAMP accumulation in COS-7 cells transfected with rat GIP receptor, while also acting as a competitive antagonist of GIP.
TP1982 Neuropeptide S(Rat)

Neuropeptide S (Rat)

Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM). Increases locomotor activity and wakefulness in mice. Also reduces anxiety-like behavior in mice.
TP2020 [Pro3]-GIP (Mouse)

GIP receptor antagonist (IC50 = 2.6μM). Inhibits GIP-stimulated insulin release from pancreatic β cells in vitro. In ob/ob mice, blocks the effects of GIP on insulin release and plasma glucose levels. Also improves intraperitoneal glucose tolerance, insul

化合物

[Pro3]-GIP (Rat)
Cat.No: TP2021
Synonym:
Target:
Neuropeptide S(Rat)
Cat.No: TP1982
Synonym: Neuropeptide S (Rat)
Target:
[Pro3]-GIP (Mouse)
Cat.No: TP2020
Synonym:
Target:
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