Cat. No. | Product Name | Target | Signaling Pathways |
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TP2021 |
[Pro3]-GIP (Rat)
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High affinity rat GIP receptor partial agonist (Kd = 13 nM). Increases cAMP accumulation in COS-7 cells transfected with rat GIP receptor, while also acting as a competitive antagonist of GIP. | |||
TP1982 |
Neuropeptide S(Rat)
Neuropeptide S (Rat) |
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Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM). Increases locomotor activity and wakefulness in mice. Also reduces anxiety-like behavior in mice. | |||
TP2020 |
[Pro3]-GIP (Mouse)
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GIP receptor antagonist (IC50 = 2.6μM). Inhibits GIP-stimulated insulin release from pancreatic β cells in vitro. In ob/ob mice, blocks the effects of GIP on insulin release and plasma glucose levels. Also improves intraperitoneal glucose tolerance, insul |