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Cat. No. Product Name Target Signaling Pathways
T40321 TNF-α-IN-6

TNF-α-IN-6 is an orally efficacious allosteric inhibitor of TNFα ( K D = 6.8 nM).
T69223 CC-1088

CC-1088 is an analog of thalidomide with potential antineoplastic activity that belongs to the functional class of agents called selective cytokine inhibitory drugs (SelCIDs). SelCIDs inhibit phosphodiesterase-4 (PDE 4), an enzyme involved in tumor necrosis factor alpha (TNF alpha) production. CC-1088 inhibits production of the cytokines vascular endothelial growth factor (VEGF) (a pro-angiogenic factor) and interleukin-6 (IL-6).
T81838 Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human)

Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human) 为一种基于FRET (荧光共振能量转移) 原理的多肽底物,通过其裂解引起的荧光强度变化来评估其活性。
T78434 Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human) TFA

Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human) TFA 为基于荧光共振能量转移的多肽底物,通过裂解引起的荧光强度变化来确定其活性。

化合物

TNF-α-IN-6
Cat.No: T40321
Synonym:
Target:
CC-1088
Cat.No: T69223
Synonym:
Target:
Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human)
Cat.No: T81838
Synonym:
Target:
Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human) TFA
Cat.No: T78434
Synonym:
Target:
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