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Cat. No. Product Name Target Signaling Pathways
T61776 TEAD-IN-2

TEAD-IN-2 is an innovative, orally bioavailable inhibitor that targets the transcriptional enhancer associate domain (TEAD). It functions by regulating TEAD through ubiquitination and/or degradation by specific compounds. This compound, TEAD-IN-2, holds potential for studying various diseases, disorders, or conditions linked to TEAD [1].
T72888 YAP-TEAD-IN-2

YAP Stem Cells
YAP-TEAD-IN-2 (化合物6)作为一种YAP-TEAD PPI抑制剂,表现出高效性,其半抑制浓度(IC50)仅为2.7 nM。
T9032 MGH-CP1

Others Others
MGH-CP1 是 TEAD2 (IC50:710 nM) 及 TEAD4 (IC50:672 nM) 自棕榈酰化抑制剂,口服有活性,可降低细胞内源性或异位表达的 TEAD 蛋白棕榈酰化水平。MGH-CP1 与 Lats1/2 缺失,是 Myc 的表达受到抑制,阻碍上皮细胞过度增殖,诱导细胞凋亡。
T76005 Super-TDU (1-31)

Super-TDU (1-31) 是 Super-TDU 的肽片段。Super-TDU (1-31) 是 YAP-TEAD 复合物的抑制剂。Super-TDU 在胃癌小鼠模型中显示出有效的抗肿瘤活性并抑制肿瘤生长。
T76005L Super-TDU (1-31) (TFA)

Super-TDU (1-31) TFA 是 Super-TDU 的肽片段。Super-TDU (1-31) TFA 是YAP-TEAD 复合物的抑制剂。Super-TDU TFA 在胃癌小鼠模型中显示出有效的抗肿瘤活性并抑制肿瘤生长。

化合物

TEAD-IN-2
Cat.No: T61776
Synonym:
Target:
YAP-TEAD-IN-2
Cat.No: T72888
Synonym:
Target: YAP
MGH-CP1
Cat.No: T9032
Synonym:
Target: Others
Super-TDU (1-31)
Cat.No: T76005
Synonym:
Target:
Super-TDU (1-31) (TFA)
Cat.No: T76005L
Synonym:
Target:
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