Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28923 |
TAS-117
TAS117,TAS 117 |
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TAS-117, a PKB/Akt inhibitor, is used potentially for the treatment of solid tumors. | |||
T62907 | TAS-117 hydrochloride | ||
TAS-117 hydrochloride 是一种选择性的、有效的、口服具有活力的别构 Akt 抑制剂,作用于 Akt1 (IC50: 4.8 nM) 、Akt2 (IC50: 1.6 nM) 和 Akt3 (IC50: 44 nM)。TAS-117 hydrochloride 能够激发抗骨髓瘤活性,增强蛋白酶体抑制诱导的致命内质网应激,可以诱导细胞凋亡和自噬。 |