Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10950 |
Dabigatran D4 hydrochloride
BIBR-953 D4 hydrochloride |
Others | Others |
Dabigatran D4 hydrochloride is deuterium-labeled dabigatran, which is a reversible and selective direct thrombin inhibitor (DTI) with a Ki value of 4.5 nM. | |||
T6295 |
Dabigatran
BIBR 953,BIBR 953ZW,达比加群 |
Thrombin | Proteases/Proteasome |
Dabigatran (BIBR 953ZW) 是一种口服抗凝剂,是一种可逆的,竞争性的直接凝血酶 (thrombin) 抑制剂,Ki=4.5 nM。它也抑制凝血酶诱导的血小板聚集 (IC50=10 nM)。 | |||
T15046 |
Dabigatran ethyl ester
Dabigatran (ethyl ester),Dabigatran ethyl ester |
Thrombin | Proteases/Proteasome |
Dabigatran ethyl ester (Dabigatran (ethyl ester)) 是新型的口服抗凝化合物和凝血酶抑制剂。 |