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Cat. No.	Product Name	Target	Signaling Pathways
T2584	Octreotide SMS 201-995,奥曲肽	Somatostatin	GPCR/G Protein
	Octreotide (SMS 201-995) 是一种有效的生长激素、胰高血糖素和胰岛素抑制剂。它主要与生长抑素 2、3 和 5 亚型受体结合，可增强 Gi 活性，降低胞内 cAMP 的产生。
T28743	Seglitide acetate MK 678,MK678,MK-678	Somatostatin	GPCR/G Protein
	Seglitide acetate (MK-678) 是一种选择性的 sst2生长抑素受体激动剂。
T9692	Paltusotine	Somatostatin	GPCR/G Protein
	Paltusotine 是一种口服有效的，非肽选择性生长抑素 2 型受体激动剂。在长效生长抑素受体配体作用后，Paltusotine 仍可维持 GH 和 IGF-1 水平。
T23073	NNC 26-9100	Others	Others
	Somatostatin sst4 receptor agonist
T24860	TC-G1003 TC G1003
	TC-G1003 is an effective agonist of the somatostatin sst2 receptor.
T69836	Paltusotine HCl
	Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.
T22487	(1R,1'S,3'R/1R,1'R,3'S)-L-054,264	Others	Others
	somatostatin sst2 receptor agonist
T27783	L-779976 L-779,976,L779,976,L779976,L 779976,L 779,976
	L-779,976 is an agonist of somatostatin receptor.
T22907	L-817,818	Others	Others
	somatostatin sst5 receptor agonist
T27787	L-797,591
	L-797,591 is a selective agonist of somatostatin receptor subtype 1.
TP2045	CH 275
	Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin release in the rat nucleus accumbens
T76544	Cyclic SSTR agonist octreotide
	Cyclic SSTR agonist octreotide 是一种 Octreotide ，可作为生长抑素受体 (SSTR) 的激动剂。
TP2124	Somatostatin 1-28
	Somatostatin receptor agonist, derived from the post-translational cleavage of prosomatostatin.
T39207	L-803087 TFA
	L-803087 TFA is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM. It displays a remarkable selectivity, being over 280-fold more preferential for the sst4 receptor compared to other somatostatin receptors. Furthermore, L-803087 TFA promotes AMPA-mediated synaptic responses in hippocampal preparations and enhances kainate-induced seizures in mice.
T32511L	L-796,778 acetate L-796,778 acetate(217480-25-6 Free base)	Somatostatin	GPCR/G Protein
	L-796,778 acetate 是一种选择性生长抑素受体激动剂，对 sst3的IC50为24nM，对sst1、sst2、sst4和sst5的IC50大于1000nM。
T11700	J-2156	Others	Others
	The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. J-2156 is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC5
T60784	SSTR4 agonist 2
	SSTR4 agonist 2 是有效的生长抑素受体亚型 4 (SSTR4) 激动剂，在 SSTR4 相关的医学疾病研究中具有潜力。SSTR4 通路抑制痛觉和炎症。
T82883	BIM-23027
	BIM-23027为高选择性sst2受体激动剂（EC50=0.32 nM），其功能效果类似生长抑素（SRIF，环状十四肽）。该化合物可促进多巴胺的释放，此过程通过Glu依赖的机制进行调控。
T75248	Pasireotide (diaspartate)
	Pasireotide (SOM230) diaspartate 是一种长效的环己肽生长激素抑制素类似物，可以提高生长抑素受体的激动剂活性，对sst1/2/3/4/5的pKi 分别为 8.2/9.0/9.1/<7.0/9.9。Pasireotide diaspartate 具有抗分泌、抗增殖和促凋亡活性。
T35669	Neuromedin C (trifluoroacetate salt)
	Neuromedin C is a bombesin-like neuropeptide that stimulates uterine smooth muscle contraction and the release of gastrin , somatostatin, and amylase in rats. Neuromedin C is a truncated form of gastrin-releasing peptide corresponding to the GRP amino acids 18-27. It inhibits GRP and bombesin binding to rat pancreatic membranes (IC50s = 0.4 and 2.2 nM, respectively), which can be reduced by sodium chloride and guanylyl imidodiphosphate . Neuromedin C induces scratching and mast cell degranulatio...
T36729	Urotensin II (goby) (trifluoroacetate salt)
	Urotensin II is a peptide vasoconstrictor and agonist of the urotensin (UT) receptor (Ki= 2.06 nM for the human recombinant receptor expressed in HEK293 cells).1It stimulates intracellular calcium mobilization in HEK293 cells expressing human and rat UT (EC50s = 0.47 and 0.78 nM, respectively) but decreases intracellular calcium concentration in goby (G. mirabilis) enterocytes when used at a concentration of 500 nM.2Urotensin II (20 mU/ml) stimulates active sodium and chloride absorption across ...

化合物

Cat.No: T2584

Synonym: SMS 201-995,奥曲肽

Target: Somatostatin

Seglitide acetate

Cat.No: T28743

Synonym: MK 678,MK678,MK-678

Target: Somatostatin

Cat.No: T9692

Target: Somatostatin

Cat.No: T23073

Target: Others

Cat.No: T24860

Synonym: TC G1003

Paltusotine HCl

Cat.No: T69836

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Cat.No: T22487

Target: Others

Cat.No: T27783

Synonym: L-779,976,L779,976,L779976,L 779976,L 779,976

Cat.No: T22907

Target: Others

Cat.No: T27787

Cat.No: TP2045

Cyclic SSTR agonist octreotide

Cat.No: T76544

Somatostatin 1-28

Cat.No: TP2124

Cat.No: T39207

L-796,778 acetate

Cat.No: T32511L

Synonym: L-796,778 acetate(217480-25-6 Free base)

Target: Somatostatin

Cat.No: T11700

Target: Others

SSTR4 agonist 2

Cat.No: T60784

Cat.No: T82883

Pasireotide (diaspartate)

Cat.No: T75248

Neuromedin C (trifluoroacetate salt)

Cat.No: T35669

Urotensin II (goby) (trifluoroacetate salt)

Cat.No: T36729

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