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Cat. No. Product Name Target Signaling Pathways
TP2352 Septide

Substance P (6-11), pyroglutamyl(6)-proline(9)-,6-Glp-9-pro-substance P (6-11)

Septide is an NK1 receptor agonist acting at a site distinct from substance P.
TP1369L [Sar9,Met(O2)11]-Substance P acetate

[Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base) 是一种速激肽 NK1 受体选择性激动剂。它是一种选择性速激肽 NK1 受体激动剂。它和 septide(每只大鼠 10-100 pmol,i.c.v.)在增加平均动脉血压 (MAP) 和心率 (HR),但它们的时间进程不同。两种激动剂都以剂量依赖性方式增加洗脸和吸鼻,而它是一种产生美容效果的化合物。
TP1369 [Sar9,Met(O2)11]-Substance P TFA(110880-55-2,free)

[Sar9,Met(O2)11]-Substance P TFA

[Sar9,Met(O2)11]-Substance P TFA is a selective tachykinin NK1 receptor agonist.[Sar9,Met(O2)11]-Substance P and septide (10-100 pmol per rat, i.c.v.) are equipotent in increasing mean arterial blood pressure (MAP) and heart rate (HR), yet they have dissi
T76402 [Glp6] Substance P (6-11)

[Glp6] Substance P (6-11)为Substance P (6-11)的一种类似物,主要通过激活大鼠膀胱中的“隔膜敏感”速激素受体,促进[3H]-单磷酸肌醇 ([3H]-IP1)的生成。

化合物

Septide
Cat.No: TP2352
Synonym: Substance P (6-11), pyroglutamyl(6)-proline(9)-,6-Glp-9-pro-substance P (6-11)
Target:
[Sar9,Met(O2)11]-Substance P acetate
Cat.No: TP1369L
Synonym: [Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base)
Target: Neurokinin receptor
[Sar9,Met(O2)11]-Substance P TFA(110880-55-2,free)
Cat.No: TP1369
Synonym: [Sar9,Met(O2)11]-Substance P TFA
Target:
[Glp6] Substance P (6-11)
Cat.No: T76402
Synonym:
Target:
TargetMol Loading
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