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Cat. No. Product Name Target Signaling Pathways
T8574 SPHINX

Others Others
SPHINX 是新一代的 SPRK1抑制剂。
T36684 Ipivivint

Ipivivint, a first-in-class, orally active and potent CDC-like kinase (CLK) inhibitor, inhibits CLK1 (IC50=1.4 μM), CLK2 (IC50=0.002 μM) and CLK3 (IC50=0.022 μM). Ipivivint reduces Wnt pathway signaling gene expression through inhibiting CLK activity and serine and arginine rich splicing factor (SRSF) phosphorylation and disrupting spliceosome activity. Ipivivint can be used for the research of cancer[1]. Ipivivint (SW480 cells; 0.01~10 μM; 1 hour) potently inhibits SRSF5/6 phosphorylation[1].Ip...

化合物

SPHINX
Cat.No: T8574
Synonym:
Target: Others
Ipivivint
Cat.No: T36684
Synonym:
Target:
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