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Cat. No. Product Name Target Signaling Pathways
TP2207 Pasireotide Acetate

Somatostatin GPCR/G Protein
Pasireotide acetate 是长效的环己肽生长激素抑制素类似物,具有抗分泌、抗增殖和促凋亡活性。它可抑制 GH、IGF-I 和 ACTH 的分泌,可用于研究肢端肥大症和库欣病。它还可以提高生长抑素受体的激动剂活性,对sst1、2、3、4、5的pKi 分别为 8.2、9.0、9.1、小于7.0 和 9.9。
T12370 Pasireotide

SOM 230,SOM 320,帕瑞肽

Others Others
Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively).
T28298 Pasireotide diaspartate

SOM-230,SOM230,trade name: Signifor,SOM 230,Signifor LAR

Pasireotide is a somatostatin analog with a 40-fold increased affinity to somatostatin receptor 5 compared to other somatostatin analogs.
T13811 Pasireotide ditrifluoroacetate

SOM230 ditrifluoroacetate,Pasireotide ditrifluoroacetate (396091-73-9 free base),Pasireotide TFA salt

Others Others
Pasireotide is a stable cyclohexapeptide somatostatin mimic.

化合物

Pasireotide Acetate
Cat.No: TP2207
Synonym:
Target: Somatostatin
Pasireotide
Cat.No: T12370
Synonym: SOM 230,SOM 320,帕瑞肽
Target: Others
Pasireotide diaspartate
Cat.No: T28298
Synonym: SOM-230,SOM230,trade name: Signifor,SOM 230,Signifor LAR
Target:
Pasireotide ditrifluoroacetate
Cat.No: T13811
Synonym: SOM230 ditrifluoroacetate,Pasireotide ditrifluoroacetate (396091-73-9 free base),Pasireotide TFA salt
Target: Others
TargetMol Loading
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