Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6875 |
Lesinurad
RDEA594,雷西那德,来司诺雷 |
OAT | Membrane transporter/Ion channel |
Lesinurad (RDEA594) 是URAT1和OAT 抑制剂。Lesinurad 用作肾转运蛋白OAT1 和OAT3 的底物,Km 分别为 0.85 和 2 μM。 | |||
T21301 |
Lesinurad sodium
Lesinurad,RDEA 594,RDEA-594,RDEA594 |
||
UNC569, the first small-molecule MER inhibitor, inhibits Mer activation and downstream signaling through ERK1/2 and AKTwith. UNC569 shows efficacy against acute lymphoblastic leukemia in vitro and in vivo. |