Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16560 |
Poloxin
|
PLK | Cell Cycle/Checkpoint |
Poloxin 是一种 polo 样激酶 1 的 ATP 非竞争性抑制剂,靶向 polo-box 结构域,IC50值约为 4.8 μM。 | |||
T25969 |
Poloxin-2
Poloxin2,Poloxin 2 |
PLK | Cell Cycle/Checkpoint |
Poloxin-2 是一种具有有效性和选择性的 Plk1 PBD 抑制剂,具有抗肿瘤活性,可降低HeLa细胞中Plk1的蛋白水平。 | |||
T16559 |
Poloxime
|
PLK | Cell Cycle/Checkpoint |
Poloxime is a hydrolysis product of poloxin and is a non-ATP-competitive Plk1 inhibitor. It also has moderate Plk1 inhibitory activity. |