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Cat. No. Product Name Target Signaling Pathways
TP1137L Pancreatic Polypeptide (human) acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Pancreatic Polypeptide (human) acetate 是一种 C 末端酰胺化的 36 个氨基酸肽,可作为神经肽 Y (NPY) Y4/Y5 受体激动剂。
TP1137 Pancreatic Polypeptide, human

Human pancreatic polypeptide

Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.
T75787 Amylin, amide, human TFA

Amylin, amide, human TFA 是一种含有37个氨基酸的胰腺多肽,与胰岛素共同分泌,对代谢和维持葡萄糖稳态具有重要作用。该化合物能够抑制胰高血糖素的分泌,延缓胃排空速度,同时作为增加饱腹感的因子。
T36864 GRP (human) (trifluoroacetate salt)

Gastrin-releasing peptide (GRP) is a neuropeptide that stimulates gastrin release. It binds to (Ki = 300 nM) and stimulates amylase secretion in rat pancreatic AR42J cells (EC50 = 0.3 nM). GRP increases proliferation of human liver carcinoma HepG2 and MHCC97H cells but does not affect the proliferation of normal HL-7702 liver cells at a concentration of 1 nM. In vivo, GRP (0.35 nmol/kg/h) increases both pancreatic exocrine secretion and pancreatic polypeptide (PP) release in rats. It dose-depend...

化合物

Pancreatic Polypeptide (human) acetate
Cat.No: TP1137L
Synonym:
Target: Neuropeptide Y Receptor
Pancreatic Polypeptide, human
Cat.No: TP1137
Synonym: Human pancreatic polypeptide
Target:
Amylin, amide, human TFA
Cat.No: T75787
Synonym:
Target:
GRP (human) (trifluoroacetate salt)
Cat.No: T36864
Synonym:
Target:
TargetMol Loading
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