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Cat. No. Product Name Target Signaling Pathways
T79067 PROTAC BTK Degrader-3

PROTACs PROTAC
PROTACBTK Degrader-3BTKPROTAC降解剂,具有效力,其在Mino细胞中BTK降解的DC50值为10.9 nM。该降解剂具有应用于研究B细胞恶性肿瘤潜力,包括慢性淋巴细胞恶性肿瘤。
T18068 Lenalidomide-PEG3-iodine

Others Others
Lenalidomide-PEG3-iodine, an E3 ligase ligand-linker conjugate, consists of a cereblon-based Lenalidomide ligand and a 3-unit polyethylene glycol (PEG) linker. This compound is utilized in creating various proteolysis targeting chimeras (PROTACs), including the highly effective PROTAC BTK degrader SJF620, which has a degradation concentration 50 (DC50) of 7.9 nM[1].

化合物

PROTAC BTK Degrader-3
Cat.No: T79067
Synonym:
Target: PROTACs
Lenalidomide-PEG3-iodine
Cat.No: T18068
Synonym:
Target: Others
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