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Cat. No. Product Name Target Signaling Pathways
T18596 PROTAC AR Degrader-4

Others Others
PROTAC AR Degrader-4 comprises a cIAP1 ligand binding group, a linker and an androgen receptor (AR) binding group. PROTAC AR Degrader-4 is an AR degrader. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs)[1].
T73726 PROTAC AR Degrader-4 TFA

PROTACAR Degrader-4 包含IAP 配体结合基团,linker 和雄激素受体 (AR) 配体结合基团。基于cIAP1的降解剂也被称为SNIPER。
T14318 ARCC-4

Others Others
ARCC-4 is an enzalutamide-based von Hippel-Lindau (VHL)-recruiting AR PROTAC and outperforms enzalutamide and it is a low-nanomolar androgen receptor (AR) degrader based on PROTAC, with a DC50 of 5 nM. ARCC-4 effectively degrades clinically relevant AR mutants associated with antiandrogen therapy[1].

化合物

PROTAC AR Degrader-4
Cat.No: T18596
Synonym:
Target: Others
PROTAC AR Degrader-4 TFA
Cat.No: T73726
Synonym:
Target:
ARCC-4
Cat.No: T14318
Synonym:
Target: Others
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