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Cat. No. | Product Name | Target | Signaling Pathways |
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T29938 |
AM-3102
KDS-5104,AM 3102,Methyl oleoylethanolamide |
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AM-3102 is an OEA analog that stimulates PPARα transcriptional activity and prolongs feeding latency. It is resistant to enzymatic hydrolysis and is as potent as OEA in enhancing transcriptional activity of PPARα and reducing food intake in free-feeding r | |||
T25366 |
Elaidyl-sulfamide
Elaidylsulfamide,ES |
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Elaidyl-sulfamide is a sulfamoyl analogue of oleoylethanolamide (OEA). ES is a lipid mediator of satiety that acts through the PPARα. | |||
T23204L |
PSN 375963 hydrochloride(388575-52-8 Free base)
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PSN 375963 hydrochloride 是一种有效的GPR119激动剂,对人和小鼠GPR119的EC50分别为 8.4 和 7.9 μM。PSN 375963 hydrochloride 表现出与内源性油酰乙醇酰胺 (OEA) 相似的效力。 | |||
T60767 |
NAAA-IN-1
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NAAA-IN-1 (Compound 1) 可用于炎症和疼痛的研究。NAAA-IN-1 是NAAA 的选择性抑制剂 (IC50 = 7 nM)。NAAA 优先水解内源性生物脂棕榈酰乙醇酰胺 (PEA) 和油酰乙醇酰胺 (OEA),是一种半胱氨酸酰胺酶。 | |||
T60378 |
NAAA-IN-2
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NAAA-IN-2 (Compound 9) 是一种有效的、选择性的NAAA 抑制剂,IC50为 50 nM。NAAA 是一种半胱氨酸酰胺酶,优先水解内源性生物脂棕榈酰乙醇酰胺 (PEA) 和油酰乙醇酰胺 (OEA)。NAAA-IN-2 在炎症和疼痛的研究中具有潜力。 | |||
T60432 |
NAAA-IN-3
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NAAA-IN-3 (Compound 17a) 是一种有效的、选择性的 NAAA 抑制剂,IC50为 50 nM。NAAA 是一种半胱氨酸酰胺酶,它优先水解内源性生物脂棕榈酰乙醇酰胺 (PEA) 和油酰乙醇酰胺 (OEA)。PEA 是核过氧化物酶体增殖物激活受体-α (PPAR-α) 的内源性激动剂,PPAR-α 是炎症和疼痛的关键调节因子。 NAAA-IN-3 的潜在作用是作为炎症和疼痛的治疗剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T12296 |
Oleoylethanolamide
油酰单乙醇胺,N-Oleoylethanolamide,Oleamide MEA,Oleic acid monoethanolamide |
Endogenous Metabolite; PPAR | DNA Damage/DNA Repair; Metabolism |
Oleoylethanolamide (N-Oleoylethanolamide) 是一种PPAR-α 的高亲和力内源性激动剂,可用于肥胖和动脉硬化的相关研究。 |