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Cat. No. Product Name Target Signaling Pathways
TP2279L Obestatin (rat) acetate

GHSR GPCR/G Protein
Obestatin (rat) acetate 是 G 蛋白偶联受体 39 (GPR39) 的内源性配体。它具有抗炎、抗心肌梗塞和抗氧化特性。 它抑制食物摄入,抑制空肠收缩,并减少体重增加。
T38470 Obestatin (human)

Obestatin (human) 是一种由 preproghrelin 经过剪切形成的G蛋白欧联实体39的内源性配体,可以剂量依赖的方式抑制进食,可用于研究肥胖。
TP2279 Obestatin(rat)

Obestatin (rat)

Others Others
Endogenous peptide that suppresses food intake and body weight-gain
T35787 Obestatin (human) (trifluoroacetate salt)

Obestatin is a 23 amino acid peptide hormone with a conserved C-terminal glycine residue and amidation site that is formed by cleavage of the ghrelin and obestatin prepropeptide.1It binds to the orphan receptor GPR39 (Kd= 1 nM) and stimulates cAMP production in CHO and HEK293 cells overexpressing human GPR39. Obestatin inhibits contraction of isolated mouse jejunum muscle strips induced by ghrelin .In vivo, obestatin (12.5-1,000 nmol/kg) suppresses food intake in a time- and dose-dependent manne...

化合物

Obestatin (rat) acetate
Cat.No: TP2279L
Synonym:
Target: GHSR
Obestatin (human)
Cat.No: T38470
Synonym:
Target:
Obestatin(rat)
Cat.No: TP2279
Synonym: Obestatin (rat)
Target: Others
Obestatin (human) (trifluoroacetate salt)
Cat.No: T35787
Synonym:
Target:
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