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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1083L Neuromedin U (rat) acetate

Others Others
Neuromedin U (rat) acetate 是一种 23 个氨基酸的脑肠肽。 Neuromedin U (NMU) 通过其在中枢神经系统中的同源受体 NMUR2 调节几种重要的生理功能,包括能量平衡、压力反应和伤害感受。
T35597 Neuromedin U-23 (rat) (trifluoroacetate salt)

Neuromedin U-23 (NMU-23) is a neuropeptide involved in diverse biological processes, including smooth muscle contraction, energy homeostasis, and nociception.1It is an agonist of neuromedin-U receptor 1 (NMUR1; EC50= 0.17 nM for the human receptor in a calcium mobilization assay using HEK293 cells) and NMUR2 (EC50= ~1.4-2 nM for arachidonic acid release in CHO cells expressing the human receptor).2,3NMU-23 (1 μM) induces contractions in isolated rat colon smooth muscle strips.4It decreases body ...
TP1083 Neuromedin U, rat

Rat neuromedin U-23,Neuromedin U (rat)

Neuromedin U,a 23-amino acid brain-gut peptide, regulates several important physiological functions through its cognate receptor NMUR2 in the central nervous system, including energy balance, stress response, and nociception.
T78004 Neuromedin U, rat TFA

Rat neuromedin U-23 TFA,Neuromedin U (rat) (TFA)

Neuromedin U, rat TFA 是一脑肠肽类化合物,含23个氨基酸,主要通过中枢神经系统内的NMUR2同源受体,调控多项生理功能,如能量平衡、应激反应及伤害感知。
T35598 Neuromedin U-25 (human) (trifluoroacetate salt)

Neuromedin U (NMU) is a neuropeptide first demonstrated to drive smooth muscle contraction.1Translated as a 174 amino acid propeptide, NMU is cleaved to different lengths in different animals. It has diverse receptor-mediated rolesin vivo, as it regulates feeding, vasoconstriction, nociception, and bone remodeling and contributes to obesity, cancer and septic shock.2,2NMU-25 is the active form of NMU in humans. It binds with high affinity to receptors on human left ventricle and coronary artery ...
TP1084 Neuromedin U, rat TFA (117505-80-3 free base)

Neuromedin U (rat) (TFA),Rat neuromedin U-23 TFA,Neuromedin U, rat TFA

Neuromedin U, rat TFA is a 23-amino acid brain-gut peptide.
T81681 Neuromedin U-25 (porcine)

Neuromedin U-25 (porcine) 是一类具有子宫刺激和升高血压作用的肽。
T81683 Neuromedin S (human)

Neuromedin S (human) 是包含33个氨基酸的神经肽,作为G 蛋白偶联受体 (GPCR) FM-4/TGR-1的内源性配体,在大脑中被鉴定,并对神经调节素 U (NMU) 受体 2 (NMUR2)调节体重稳态具有调控作用。
TP1980 Neuromedin S(rat)

Neuromedin S (rat)

Potent, endogenous neuromedin U receptor agonist (EC50 values are 65 and 91 pM at NMU1 and NMU2 respectively). Induces phase shifts in the circadian rhythm of locomotor activity following i.c.v. administration. Potent endogenous anorexigenic peptide.

化合物

Neuromedin U (rat) acetate
Cat.No: TP1083L
Synonym:
Target: Others
Neuromedin U-23 (rat) (trifluoroacetate salt)
Cat.No: T35597
Synonym:
Target:
Neuromedin U, rat
Cat.No: TP1083
Synonym: Rat neuromedin U-23,Neuromedin U (rat)
Target:
Neuromedin U, rat TFA
Cat.No: T78004
Synonym: Rat neuromedin U-23 TFA,Neuromedin U (rat) (TFA)
Target:
Neuromedin U-25 (human) (trifluoroacetate salt)
Cat.No: T35598
Synonym:
Target:
Neuromedin U, rat TFA (117505-80-3 free base)
Cat.No: TP1084
Synonym: Neuromedin U (rat) (TFA),Rat neuromedin U-23 TFA,Neuromedin U, rat TFA
Target:
Neuromedin U-25 (porcine)
Cat.No: T81681
Synonym:
Target:
Neuromedin S (human)
Cat.No: T81683
Synonym:
Target:
Neuromedin S(rat)
Cat.No: TP1980
Synonym: Neuromedin S (rat)
Target:
Cat. No. Product Name Target Signaling Pathways
T8035 3'-Methoxyflavonol

NMU2R Neuroscience
3'-Methoxyflavonol 是一种神经介肽 U 2 受体的选择性激动剂。

天然产物

3'-Methoxyflavonol
Cat.No: T8035
Synonym:
Target: NMU2R
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