Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T71749 |
SF-22
|
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
SF-22 是一种可透过血脑屏障的神经肽 Y 受体(Y2R) 拮抗剂,具有潜在抗炎活性,可用于研究神经系统紊乱带来的疾病。 | |||
T29171 |
Y2 Antagonist 36
|
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Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2. | |||
T71091 |
Y2-Antagonist-2
|
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Y2-Antagonist-2 is a novel, selective, soluble non-peptidic NPY Y2 receptor antagonist with enhanced CNS exposure. | |||
T10921 |
CYM 9484
|
Others | Others |
CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with IC50 value of 19 nM. | |||
T14572 |
BIIE-0246
AR-H 053591 |
Others | Others |
BIIE-0246 is a potent and highly selective non-peptide neuropeptide Y (NPY) Y2 receptor antagonist. With an IC50 of 15 nM. | |||
T36481 | BIIE 0246 hydrochloride | ||
Potent, selective and competitive nonpeptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM). Displays > 650-fold selectivity for NPY Y2 over Y1, Y4 and Y5 receptors. Active in vivo. | |||
T41188 |
BIBP 3226 trifluoroacetate
|
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BIBP 3226 trifluoroacetate is a mixed non-peptide neuropeptide Y Y1(NPY Y1) and neuropeptide FF (NPFF) receptor antagonist (Kivalues are 1.1, 79, 108, > 1000, > 1000 and >1000 for rNPY Y1, hNPFF2, rNPFF, rNPY Y2, rNPY Y4and rNPY Y5respectively). Produces an anxiogenic-like effect in rats following i.c.v. administration. |