Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1425 |
Motilin (26-47), human, porcine
胃动素 (人类,猪) |
Motilin Receptor | GPCR/G Protein |
Motilin (26-47), human, porcine 是内源性 motilin 受体的激动剂,在中国仓鼠卵巢细胞中,Ki 值和EC50值分别为 2.3 和 0.3 nM。 | |||
T11508L |
Camicinal hydrochloride
GSK962040 hydrochloride |
Others; Motilin Receptor | GPCR/G Protein; Others |
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。 | |||
T11508 |
Camicinal
GSK962040 |
Others | Others |
Camicinal is a selective motilin receptor agonist (pEC50: 7.9). | |||
T15946 | MA-2029 | Others | Others |
MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 may be useful for gastrointestinal disorders associated with disturbed g | |||
T76359 |
[Nle13]-Motilin
|
||
[Nle13]-Motilin 是一种胃动素 (motilin) 类似物,可作为胃动素受体 motilin receptor 激动剂。 | |||
T27584 |
Idremcinal
EM574,EM 574,EM-574 |
||
Idremcinal is a motilin receptor agonist. | |||
T29174 |
YIL781 hydrochloride
YIL 781,YIL-781,YIL781 HCl,YIL781 |
||
YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM). |