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Cat. No. | Product Name | Target | Signaling Pathways |
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TP1425 |
Motilin (26-47), human, porcine
胃动素 (人类,猪) |
Motilin Receptor | GPCR/G Protein |
Motilin (26-47), human, porcine 是内源性 motilin 受体的激动剂,在中国仓鼠卵巢细胞中,Ki 值和EC50值分别为 2.3 和 0.3 nM。 | |||
TP1098 |
Motilin, canine
Motilin (canine) |
||
Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist. | |||
T78563 |
[Leu13]-Motilin
KW-5139 |
Motilin Receptor | GPCR/G Protein |
[Leu13]-Motilin (KW-5139) 为motilin类似物,能够刺激家兔胃肠运动,并在体外以浓度依赖性方式引起胃窦、十二指肠、空肠、回肠以及降结肠的收缩。 | |||
T76359 |
[Nle13]-Motilin
|
||
[Nle13]-Motilin 是一种胃动素 (motilin) 类似物,可作为胃动素受体 motilin receptor 激动剂。 | |||
T11508L |
Camicinal hydrochloride
GSK962040 hydrochloride |
Others; Motilin Receptor | GPCR/G Protein; Others |
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。 | |||
T11508 |
Camicinal
GSK962040 |
Others | Others |
Camicinal is a selective motilin receptor agonist (pEC50: 7.9). | |||
T15946 | MA-2029 | Others | Others |
MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 is a selective and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 may be useful for gastrointestinal disorders associated with disturbed g | |||
T27584 |
Idremcinal
EM574,EM 574,EM-574 |
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Idremcinal is a motilin receptor agonist. | |||
T70464 |
Mitemcinal
|
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Mitemcinal is a motilin agonist. | |||
T29174 |
YIL781 hydrochloride
YIL 781,YIL-781,YIL781 HCl,YIL781 |
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YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM). | |||
T75861 |
ANQ-11125 TFA
|
||
ANQ-11125 TFA 是一种有效的、选择性胃动素拮抗剂,pKd 值为 8.24。ANQ-11125 TFA 在体外阻断 motilide 引起的收缩。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-04207 |
Motilin Protein, Human, Recombinant (His)
MLN,Motilin |
Human | HEK293 Cells |
MLN (Motilin) is a Protein Coding gene. 3 alternatively spliced human isoforms have been reported. This gene encodes a small peptide hormone that is secreted by cells of the small intestine to regulate gastrointestinal contractions and motility. The encoded protein belongs to the motilin family. Proteolytic processing of the secreted protein produces the mature peptide and a byproduct referred to as motilin-associated peptide (MAP). MLN plays an important role in the regulation of Interdigestive... | |||
TMPH-01922 |
Promotilin Protein, Human, Recombinant (GST & His & Myc)
|
Human | E. coli |
Promotilin Protein, Human, Recombinant (GST & His & Myc) is expressed in E. coli. |